SCHEMBL7050895

SCHEMBL7050895

CCCc1cc2c(N3CCN(C(C=O)c4ccccc4)C[C@@H]3C)nc(C)nc2s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.38
CNR2 P34972 4/20 0.37
CNR1 P21554 2/20 0.36
CYP2D6 P10635 1/20 0.36
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 4/20 0.36
HPGD P15428 3/20 0.36
MAPK1 P28482 2/20 0.36
TSHR P16473 2/20 0.36
LMNA P02545 1/20 0.36
HSD17B10 Q99714 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
POLB P06746 1/20 0.34
USP7 Q93009 1/20 0.33
HTT P42858 3/20 0.33
GPR55 Q9Y2T6 1/20 0.32
P2RY12 Q9H244 3/20 0.32
NPSR1 Q6W5P4 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7048493 0.80 SMN1; SMN2 (0.51) KDM4EALDH1A1MAPK1TSHRLMNA
SCHEMBL7054382 0.80 SMN1; SMN2 (0.51) KDM4EALDH1A1MAPK1TSHRLMNA
SCHEMBL7046759 0.79 HTR6 (0.60) HTR6CNR2CNR1CYP2D6KDM4E
SCHEMBL5851706 0.78 HTR6 (0.43) HTR6CNR2CNR1CYP2D6KDM4E
SCHEMBL7052172 0.77 HTR6 (0.31) HTR6
SCHEMBL7053533 0.75 HTT (0.56) KDM4EALDH1A1TSHRLMNASMN1; SMN2
SCHEMBL7055758 0.73 TP53 (0.45) HTR6TSHRSMN1; SMN2MEN1KMT2A
SCHEMBL7051621 0.70 TP53 (0.47) HTR6TSHRSMN1; SMN2MEN1KMT2A
SCHEMBL7047637 0.70 TP53 (0.45) HTR6TSHRSMN1; SMN2MEN1KMT2A
SCHEMBL7050247 0.69 P2RY12 (0.46) HTR6TSHRSMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003022214-A2 PIPERAZINE AND HOMOPIPERAZINE COMPOUNDS MILLENNIUM PHARMACEUTICALS, INC. (US) 2003-03-20 WO disclosed