SCHEMBL7046759

SCHEMBL7046759

CCc1cc2c(N3CCN(C(C=O)c4ccccc4)CC3)nc(C)nc2s1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.60
CNR2 P34972 4/20 0.49
CNR1 P21554 2/20 0.49
CYP2D6 P10635 1/20 0.49
MEN1 O00255 4/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
KMT2A Q03164 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TSHR P16473 2/20 0.47
HTT P42858 2/20 0.47
POLB P06746 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HPGD P15428 2/20 0.46
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.46
HSD17B10 Q99714 1/20 0.46
P2RY12 Q9H244 9/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7051621 0.90 TP53 (0.47) HTR6MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL7050247 0.89 P2RY12 (0.46) HTR6MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL7055819 0.89 TP53 (0.46) HTR6MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL7047637 0.88 TP53 (0.45) HTR6MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL7055758 0.88 TP53 (0.45) HTR6MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL7050374 0.88 TP53 (0.45) HTR6MEN1KDM4EALDH1A1KMT2A
SCHEMBL7048623 0.85 HTT (0.67) MEN1KDM4EALDH1A1KMT2ASMN1; SMN2
SCHEMBL7047651 0.79 HTT (0.45) MEN1KDM4EALDH1A1KMT2ASMN1; SMN2
SCHEMBL7050895 0.79 HTR6 (0.38) HTR6CNR2CNR1CYP2D6MEN1
SCHEMBL7053533 0.78 HTT (0.56) MEN1KDM4EALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003022214-A2 PIPERAZINE AND HOMOPIPERAZINE COMPOUNDS MILLENNIUM PHARMACEUTICALS, INC. (US) 2003-03-20 WO disclosed