SCHEMBL7051606

SCHEMBL7051606

Cc1c(-c2ccccc2)oc2c(C(=O)NCCCN3CCN(c4cc(Cl)ccc4O)CC3)cccc2c1=O

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.72
ADRA1A P35348 6/20 0.72
ADRA1D P25100 5/20 0.72
ADRA1B P35368 5/20 0.72
LMNA P02545 2/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
ALDH1A1 P00352 1/20 0.60
MAPT P10636 1/20 0.60
NPSR1 Q6W5P4 1/20 0.60
HTR2A P28223 6/20 0.53
HTR2C P28335 6/20 0.53
SLC6A4 P31645 6/20 0.53
DRD3 P35462 3/20 0.51
KCNH2 Q12809 3/20 0.51
KDM4E B2RXH2 1/20 0.51
CYP1A2 P05177 1/20 0.51
CHRM2 P08172 1/20 0.51
CYP3A4 P08684 1/20 0.51
ADRA2A P08913 1/20 0.51
ADORA3 P0DMS8 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7051331 0.91 HTR1A (0.81) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8875520 0.91 HTR1A (0.84) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8876351 0.89 HTR1A (0.81) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8876429 0.89 HTR1A (0.71) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8875778 0.88 HTR1A (0.73) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7050780 0.87 HTR1A (0.55) HTR1AADRA1AADRA1DADRA1BSMN1; SMN2
SCHEMBL7054044 0.87 HTR1A (0.69) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL8875767 0.87 HTR1A (0.77) HTR1AADRA1AADRA1DADRA1BLMNA
SCHEMBL7052255 0.86 HTR1A (0.68) HTR1AADRA1AADRA1DADRA1BLMNA
Hydrochloric Acid SCHEMBL7054302 0.86 HTR1A (0.67) HTR1AADRA1AADRA1DADRA1BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US claimed
EP-1222183-B1 BENZOPYRAN DERIVATIVES RECORDATI CHEM PHARM (IT) 2003-04-23 EP disclosed
US-6403594-B1 UROGENTIAL INFECTIONS, ETC RECORDATI, S.A. CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 2002-06-11 US disclosed