SCHEMBL7052827

SCHEMBL7052827

CC(=O)ON=C1C(=O)C(=O)Nc2cc(C(F)(F)F)cc(Cl)c21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.38
UCHL3 P15374 3/20 0.32
UCHL1 P09936 3/20 0.32
CCNB2 O95067 1/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
CCNB3 Q8WWL7 1/20 0.31
JUN P05412 2/20 0.31
NFKB1 P19838 2/20 0.31
NFKB2 Q00653 2/20 0.31
RELA Q04206 2/20 0.31
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
GABRA1 P14867 1/20 0.31
GABRB1 P18505 1/20 0.31
GABRG2 P18507 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7050452 0.92 CES1 (0.38) CES1UCHL3UCHL1CCNB2CDK1
SCHEMBL7056837 0.87 ALDH1A1 (0.30) ALDH1A1MAPTHPGDALOX15HSD17B10
SCHEMBL7047393 0.86 CES1 (0.54) CES1UCHL3UCHL1CCNB2CDK1
SCHEMBL7049367 0.86 NOTUM (0.32) CES1CCNB2CDK1CCNB1GSK3A
SCHEMBL7054180 0.83 HPGD (0.37) CES1ALDH1A1MAPTMAPK1HPGD
SCHEMBL7048278 0.81 GALR3 (0.32) ALDH1A1MAPTHPGDALOX15HSD17B10
SCHEMBL8871331 0.81 CES1 (0.45) CES1JUNNFKB1NFKB2RELA
SCHEMBL8871333 0.81 CES1 (0.45) CES1JUNNFKB1NFKB2RELA
SCHEMBL7053378 0.80 CES1 (0.39) CES1UCHL3UCHL1CCNB2CDK1
SCHEMBL7051913 0.80 GALR3 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706396-B1 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE-3 OR 4-OXIMES AND USE OREGON STATE (US) 2003-05-02 EP disclosed
US-5652368-A NERVOUS SYSTEM DISORDERS, ALZHEIMER'S DISEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-07-29 US disclosed
US-5475007-A Preventing convulsions THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-12 US disclosed