SCHEMBL7053378

SCHEMBL7053378

CC(=O)ON=C1C(=O)C(=O)Nc2cc(Cl)c(Cl)c(Cl)c21

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES1 P23141 5/20 0.39
UCHL3 P15374 4/20 0.34
UCHL1 P09936 4/20 0.34
CCNB2 O95067 2/20 0.33
CDK1 P06493 2/20 0.33
CCNB1 P14635 2/20 0.33
GSK3A P49840 2/20 0.33
GSK3B P49841 2/20 0.33
CDK5 Q00535 2/20 0.33
CDK5R1 Q15078 2/20 0.33
CCNB3 Q8WWL7 2/20 0.33
TGM2 P21980 1/20 0.32
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7048302 0.90 CES1 (0.36) CES1UCHL3UCHL1CCNB2CDK1
SCHEMBL7047393 0.85 CES1 (0.54) CES1UCHL3UCHL1CCNB2CDK1
SCHEMBL7052308 0.85 TSHR (0.36) CES1UCHL3UCHL1CCNB2CDK1
SCHEMBL7050080 0.85 CES1 (0.33) CES1UCHL3UCHL1CCNB2CDK1
SCHEMBL7051545 0.82 KMT2A (0.39) CES1TGM2ALDH1A1LMNAMAPT
SCHEMBL7050695 0.81 CES1 (0.53) CES1UCHL3UCHL1CCNB2CDK1
SCHEMBL7052827 0.80 CES1 (0.38) CES1UCHL3UCHL1CCNB2CDK1
SCHEMBL7051894 0.79 UCHL3 (0.38) CES1UCHL3UCHL1CCNB2CDK1
SCHEMBL7048414 0.79 CES1 (0.46) CES1TGM2ALDH1A1
SCHEMBL7048416 0.79 CES1 (0.46) CES1TGM2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706396-B1 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE-3 OR 4-OXIMES AND USE OREGON STATE (US) 2003-05-02 EP disclosed
US-5652368-A NERVOUS SYSTEM DISORDERS, ALZHEIMER'S DISEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-07-29 US disclosed
US-5475007-A Preventing convulsions THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-12 US disclosed