SCHEMBL7052957

SCHEMBL7052957

O=C1Nc2ccccc2C(=O)C1=NOC(=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.50
ALDH1A1 P00352 6/20 0.50
HPGD P15428 2/20 0.50
F2 P00734 1/20 0.50
ATM Q13315 1/20 0.50
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
MAPT P10636 5/20 0.47
LRRK2 Q5S007 4/20 0.47
MEN1 O00255 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
LMNA P02545 1/20 0.47
IDO1 P14902 1/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
AGTR1 P30556 1/20 0.45
MAPK1 P28482 2/20 0.44
KDR P35968 1/20 0.42
PLA2G1B P04054 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7055896 0.89 KMT2A (0.50) KMT2AALDH1A1HPGDF2ATM
SCHEMBL7049532 0.83 KMT2A (0.43) KMT2AALDH1A1HPGDF2ATM
SCHEMBL7051552 0.83 CES1 (0.47) KMT2AALDH1A1HPGDF2ATM
SCHEMBL7055054 0.83 KMT2A (0.50) KMT2AALDH1A1MAOAMAOBMAPT
SCHEMBL10624339 0.79 ALDH1A1 (0.57) KMT2AALDH1A1HPGDF2ATM
SCHEMBL7054941 0.78 KMT2A (0.38) KMT2AALDH1A1HPGDF2ATM
SCHEMBL7051548 0.77 CES1 (0.48) KMT2AALDH1A1HPGDF2ATM
SCHEMBL7054751 0.77 KMT2A (0.38) KMT2AALDH1A1HPGDF2ATM
SCHEMBL7050457 0.77 KMT2A (0.38) KMT2AALDH1A1HPGDF2ATM
SCHEMBL7052934 0.76 KMT2A (0.41) KMT2AALDH1A1HPGDF2ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706396-B1 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE-3 OR 4-OXIMES AND USE OREGON STATE (US) 2003-05-02 EP disclosed
US-5475007-A Preventing convulsions THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-12 US disclosed