SCHEMBL7053388

SCHEMBL7053388

CC(=O)ON=C1C(=O)C(=O)Nc2cc(Br)c(Br)cc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 3/20 0.44
BCHE P06276 1/20 0.44
AGTR1 P30556 1/20 0.34
TGM2 P21980 4/20 0.33
CA1 P00915 3/20 0.33
CCNB2 O95067 3/20 0.33
CDK1 P06493 3/20 0.33
CCNB1 P14635 3/20 0.33
CCNB3 Q8WWL7 3/20 0.33
CA12 O43570 2/20 0.33
CA9 Q16790 2/20 0.33
UCHL1 P09936 2/20 0.33
UCHL3 P15374 2/20 0.33
GSK3A P49840 2/20 0.33
GSK3B P49841 2/20 0.33
CDK5 Q00535 2/20 0.33
CDK5R1 Q15078 2/20 0.33
CA2 P00918 2/20 0.33
AURKB Q96GD4 2/20 0.32
AURKC Q9UQB9 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7052316 0.89 CES1 (0.44) CES1BCHEAGTR1TGM2CA1
SCHEMBL7053093 0.86 CES1 (0.38) CES1BCHEAGTR1TGM2CCNB2
SCHEMBL7050695 0.83 CES1 (0.53) CES1BCHETGM2CCNB2CDK1
SCHEMBL7052947 0.81 KMT2A (0.43) CES1BCHECCNB2CDK1CCNB1
SCHEMBL7054935 0.77 CES1 (0.49) CES1BCHEAGTR1TGM2CA1
SCHEMBL7054937 0.77 CES1 (0.49) CES1BCHEAGTR1TGM2CA1
SCHEMBL7051088 0.77 KMT2A (0.50) AGTR1TGM2ALDH1A1LMNAPOLB
SCHEMBL7053898 0.77 TGM2 (0.33) CES1TGM2
SCHEMBL7055737 0.76 CES1 (0.38) CES1BCHETGM2CCNB2CDK1
SCHEMBL7053901 0.76 CES1 (0.38) CES1TGM2CCNB2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0706396-B1 1,2,3,4-TETRAHYDROQUINOLINE-2,3,4-TRIONE-3 OR 4-OXIMES AND USE OREGON STATE (US) 2003-05-02 EP disclosed
US-5652368-A NERVOUS SYSTEM DISORDERS, ALZHEIMER'S DISEASE THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-07-29 US disclosed
US-5475007-A Preventing convulsions THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-12 US disclosed