SCHEMBL7053662

SCHEMBL7053662

COC(=O)COc1ccc(C(CC(=O)NCc2ccc(OC)cc2)NS(=O)(=O)c2ccccc2)cc1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47
POLB P06746 2/20 0.46
TP53 P04637 1/20 0.46
SGMS1 Q86VZ5 1/20 0.45
PLA2G1B P04054 1/20 0.45
ATG4B Q9Y4P1 1/20 0.45
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.43
BDKRB1 P46663 2/20 0.43
BDKRB2 P30411 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
EGFR P00533 1/20 0.41
ERBB2 P04626 1/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650912 0.94 ALDH1A1 (0.47) ALDH1A1MMP2MMP9POLBTP53
SCHEMBL4651316 0.94 ALDH1A1 (0.48) ALDH1A1MMP2MMP9POLBTP53
SCHEMBL7050019 0.85 ALDH1A1 (0.54) ALDH1A1POLBTP53SGMS1KMT2A
SCHEMBL4650872 0.83 ALDH1A1 (0.60) ALDH1A1POLBTP53KMT2AMEN1
SCHEMBL7053651 0.82 POLB (0.51) ALDH1A1MMP2MMP9POLBSGMS1
SCHEMBL4650271 0.78 BDKRB1 (0.45) ALDH1A1MMP2MMP9POLBKDM4E
SCHEMBL4651379 0.77 ALDH1A1 (0.58) ALDH1A1POLBLMNAKMT2AMEN1
SCHEMBL4650322 0.77 ALDH1A1 (0.48) ALDH1A1POLBTP53PLA2G1BATG4B
SCHEMBL7050666 0.76 POLB (0.40) ALDH1A1POLBKDM4EKMT2A
SCHEMBL4650884 0.76 PTPN1 (0.49) ALDH1A1MMP2MMP9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1301474-A2 TYROSINE DERIVATIVES AS PHOSPHATASE INHIBITORS Array Biopharma Inc. (US) 2003-04-16 EP disclosed
WO-2002004412-A2 TYROSINE DERIVATIVES AS PHOSPHATASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2002-01-17 WO disclosed