SCHEMBL7053717

SCHEMBL7053717

Cc1c(Br)ccc(N2CCN(CCCCNC(=O)c3cnc4ccccc4c3)CC2)c1C

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 17/20 0.71
DRD2 P14416 17/20 0.71
HTR1A P08908 9/20 0.71
HTR2A P28223 8/20 0.71
HTR2C P28335 7/20 0.71
ADRA1A P35348 8/20 0.58
ADRA2A P08913 5/20 0.56
ADRA1D P25100 3/20 0.56
ADRA1B P35368 3/20 0.56
ADRA2B P18089 2/20 0.56
ADRA2C P18825 2/20 0.56
HRH1 P35367 2/20 0.56
KCNH2 Q12809 1/20 0.56
DRD4 P21917 3/20 0.52
DRD1 P21728 2/20 0.51
HTR2B P41595 2/20 0.51
MEN1 O00255 1/20 0.51
LMNA P02545 1/20 0.51
TP53 P04637 1/20 0.51
CYP1A2 P05177 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4533987 0.80 SLC6A4 (0.72) DRD3DRD2HTR1AHTR2AHTR2C
SCHEMBL7058620 0.80 DRD2 (0.69) DRD3DRD2HTR1AHTR2AHTR2C
SCHEMBL7055333 0.79 DRD2 (0.70) DRD3DRD2HTR1AHTR2AHTR2C
SCHEMBL4521349 0.78 DRD3 (0.73) DRD3DRD2HTR1AHTR2AHTR2C
SCHEMBL4519092 0.77 DRD3 (1.00) DRD3DRD2HTR1AHTR2AHTR2C
SCHEMBL28071107 0.74 PLD1 (0.62) DRD3DRD2HTR1AHTR2AHTR2C
SCHEMBL5020897 0.72 HDAC3 (0.61) DRD3DRD2HTR1AHTR2AHTR2C
SCHEMBL7059254 0.72 DRD3 (0.65) DRD3DRD2HTR1AHTR2AHTR2C
SCHEMBL7057784 0.72 DRD2 (0.48) DRD3DRD2HTR1AHTR2AHTR2C
Hydrochloric Acid SCHEMBL7534187 0.72 DRD2 (0.93) DRD3DRD2HTR1AHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028728-A1 4-(4-SUBSTITUTED PIPERAZINYL-1YL)-BUTYLCARBOXAMIDES AS D3 DOPAMINE SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed