SCHEMBL7058620

SCHEMBL7058620

COc1cc(-c2ccccc2)ccc1N1CCN(CCCCNC(=O)c2cnc3ccccc3c2)CC1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 17/20 0.69
DRD3 P35462 15/20 0.69
HTR1A P08908 9/20 0.69
HTR2A P28223 7/20 0.69
HTR2C P28335 7/20 0.69
DRD4 P21917 7/20 0.66
KCNH2 Q12809 1/20 0.66
SLC6A2 P23975 2/20 0.62
SLC6A4 P31645 2/20 0.62
ADRA2A P08913 4/20 0.61
HTR2B P41595 4/20 0.61
DRD1 P21728 2/20 0.61
ADRA1D P25100 2/20 0.61
ADRA1A P35348 2/20 0.61
ADRA1B P35368 2/20 0.61
CYP1A2 P05177 2/20 0.61
MEN1 O00255 1/20 0.61
LMNA P02545 1/20 0.61
TP53 P04637 1/20 0.61
CYP3A4 P08684 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4521349 0.81 DRD3 (0.73) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL7053717 0.80 DRD3 (0.71) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL17194866 0.80 DRD2 (1.00) DRD2DRD3HTR1ADRD4KCNH2
SCHEMBL1543274 0.80 DRD2 (0.65) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL7052933 0.79 DRD2 (0.66) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL7056485 0.78 DRD2 (0.64) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL4533987 0.78 SLC6A4 (0.72) DRD2DRD3HTR1AHTR2AHTR2C
SCHEMBL14006129 0.77 DRD2 (0.69) DRD2DRD3HTR1AHTR2AHTR2C
Bp-897 SCHEMBL2125882 0.77 DRD2 (1.00) DRD2DRD3HTR1AHTR2AHTR2C
Bp-897 SCHEMBL29382551 0.77 DRD2 (1.00) DRD2DRD3HTR1AHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028728-A1 4-(4-SUBSTITUTED PIPERAZINYL-1YL)-BUTYLCARBOXAMIDES AS D3 DOPAMINE SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed