SCHEMBL7053778

SCHEMBL7053778

O=C(NCCCCN1CCN(c2cccc(C(F)(F)F)c2)CC1)c1ccc2[nH]ccc2c1

nearest known ligand 0.76

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 13/20 0.76
DRD3 P35462 13/20 0.76
ADRA1A P35348 7/20 0.76
HTR1A P08908 4/20 0.68
HTR2A P28223 4/20 0.68
HTR2C P28335 1/20 0.68
TRPV1 Q8NER1 1/20 0.53
ADRA2A P08913 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
ADRA1D P25100 1/20 0.51
HRH1 P35367 1/20 0.51
ADRA1B P35368 1/20 0.51
KCNH2 Q12809 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7058141 0.83 DRD2 (0.53) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL7058045 0.82 DRD2 (0.75) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL4525593 0.81 DRD2 (1.00) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL7056412 0.80 DRD2 (0.73) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL7056355 0.80 DRD2 (0.73) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL7056313 0.80 DRD3 (0.73) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL7056222 0.79 DRD3 (0.75) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL30389513 0.78 DRD3 (0.74) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL27014500 0.78 DRD3 (0.74) DRD2DRD3ADRA1AHTR1AHTR2A
SCHEMBL14006088 0.77 HDAC1 (0.58) DRD2DRD3ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028728-A1 4-(4-SUBSTITUTED PIPERAZINYL-1YL)-BUTYLCARBOXAMIDES AS D3 DOPAMINE SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed