SCHEMBL7056313

SCHEMBL7056313

N#Cc1ccc(C(=O)NCCCCN2CCN(c3cccc(C(F)(F)F)c3)CC2)cc1

nearest known ligand 0.73

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 13/20 0.73
DRD2 P14416 12/20 0.73
ADRA1A P35348 2/20 0.73
DRD4 P21917 1/20 0.62
HTR1A P08908 3/20 0.62
HTR2A P28223 3/20 0.62
HTR2C P28335 1/20 0.62
KCNH2 Q12809 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7056412 0.85 DRD2 (0.73) DRD3DRD2ADRA1ADRD4HTR1A
SCHEMBL7056355 0.85 DRD2 (0.73) DRD3DRD2ADRA1ADRD4HTR1A
SCHEMBL7052681 0.84 DRD3 (0.67) DRD3DRD2ADRA1ADRD4
SCHEMBL7058045 0.83 DRD2 (0.75) DRD3DRD2ADRA1AHTR1AHTR2A
SCHEMBL7055846 0.82 DRD3 (0.73) DRD3DRD2ADRA1ADRD4KCNH2
SCHEMBL7052921 0.81 DRD2 (0.70) DRD3DRD2ADRA1AHTR1AHTR2A
SCHEMBL7050873 0.81 DRD2 (0.67) DRD3DRD2ADRA1ADRD4HTR1A
SCHEMBL7056586 0.81 DRD2 (0.69) DRD3DRD2ADRA1AHTR1AHTR2A
SCHEMBL7053778 0.80 DRD2 (0.76) DRD3DRD2ADRA1AHTR1AHTR2A
SCHEMBL7058039 0.80 DRD3 (0.79) DRD3DRD2ADRA1ADRD4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028728-A1 4-(4-SUBSTITUTED PIPERAZINYL-1YL)-BUTYLCARBOXAMIDES AS D3 DOPAMINE SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed