SCHEMBL7054843

SCHEMBL7054843

CC(=O)OCCC#Cc1cccnc1

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 5/20 0.55
CHRNA4 P43681 5/20 0.55
CYP2A6 P11509 4/20 0.51
CYP2C9 P11712 3/20 0.51
CYP2B6 P20813 3/20 0.51
CYP2C19 P33261 3/20 0.51
CYP3A4 P08684 3/20 0.50
CYP2E1 P05181 2/20 0.50
CYP2D6 P10635 2/20 0.50
CYP1A2 P05177 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CYP2C8 P10632 1/20 0.49
FFAR1 O14842 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
GRM5 P41594 1/20 0.41
ERN1 O75460 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7051816 0.82 FFAR1 (0.40) CYP3A4CYP1A2MEN1KMT2AFFAR1
SCHEMBL7055462 0.82 ALDH1A1 (0.46) CYP2C9CYP2C19CYP3A4CYP2D6CYP1A2
SCHEMBL6133051 0.77 CHRNB2 (0.55) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL4065112 0.75 CHRNB2 (0.63) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL14085289 0.75 CHRNB2 (0.69) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL5376053 0.75 CHRNB2 (0.63) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL45751 0.74 KMT2A (0.42) KMT2ALMNA
SCHEMBL7453172 0.74 CHRNB2 (0.51) CHRNB2CHRNA4CYP2A6CYP2C9CYP2B6
SCHEMBL6689389 0.74 ALDH1A1 (0.50) MEN1KMT2AFFAR1LMNA
SCHEMBL46934 0.73 ALDH1A1 (0.38) CYP3A4CYP1A2MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303615-A2 FERMENTATION PROCESS FOR EPOTHILONES Kosan Biosciences, Inc. (US) 2003-04-23 EP disclosed
WO-2002008440-A2 FERMENTATION PROCESS FOR EPOTHILONES KOSAN BIOSCIENCES, INC. (US) 2002-01-31 WO disclosed