SCHEMBL7057178

SCHEMBL7057178

CNC(=O)c1cc(-c2ccc(F)cc2)sc1NC(N)=O

nearest known ligand 0.76

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 14/20 0.76
MAP4K4 O95819 1/20 0.76
IKBKB O14920 4/20 0.76
JAK2 O60674 2/20 0.76
MEN1 O00255 1/20 0.76
EIF2AK2 P19525 1/20 0.76
KMT2A Q03164 1/20 0.76
TDP1 Q9NUW8 1/20 0.76
HDAC6 Q9UBN7 1/20 0.76
CDK2AP1 O14519 1/20 0.60
JAK3 P52333 1/20 0.56
KDM4E B2RXH2 1/20 0.51
NPC1 O15118 1/20 0.51
ALDH1A1 P00352 1/20 0.51
HPGD P15428 1/20 0.51
RAB9A P51151 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7055932 0.88 CHEK1 (0.59) CHEK1MAP4K4IKBKBJAK2MEN1
SCHEMBL7055087 0.88 IKBKB (0.78) CHEK1MAP4K4IKBKBJAK2MEN1
Fluorobenzene SCHEMBL27676739 0.87 CHEK1 (0.71) CHEK1MAP4K4IKBKBJAK2MEN1
SCHEMBL7055226 0.86 CHEK1 (1.00) CHEK1MAP4K4IKBKBJAK2CDK2AP1
SCHEMBL717369 0.86 IKBKB (1.00) CHEK1IKBKBJAK2MEN1EIF2AK2
SCHEMBL3086954 0.85 IKBKB (0.82) CHEK1MAP4K4IKBKBJAK2MEN1
SCHEMBL28374187 0.84 IKBKB (0.76) CHEK1MAP4K4IKBKBJAK2MEN1
SCHEMBL5898657 0.82 IKBKB (0.76) CHEK1MAP4K4IKBKBJAK2MEN1
SCHEMBL7054417 0.81 TUBB4A (0.58) CHEK1MAP4K4IKBKBJAK2MEN1
SCHEMBL4215417 0.80 CHEK1 (0.70) CHEK1MAP4K4IKBKBJAK2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003029241-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO claimed
WO-2003029241-A1 CHK1 KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2003-04-10 WO disclosed