SCHEMBL7057729

SCHEMBL7057729

COc1cc(Br)ccc1N1CCN(CCCCNC(=O)c2cc3c(cn2)[nH]c2ccccc23)CC1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.59
DRD3 P35462 9/20 0.59
DRD4 P21917 6/20 0.59
FAAH O00519 1/20 0.56
HTR2A P28223 2/20 0.56
HTR1A P08908 1/20 0.56
MEN1 O00255 1/20 0.54
POLB P06746 1/20 0.54
RAB9A P51151 1/20 0.54
KMT2A Q03164 1/20 0.54
HDAC3 O15379 3/20 0.53
HDAC4 P56524 3/20 0.53
HDAC1 Q13547 3/20 0.53
HDAC7 Q8WUI4 3/20 0.53
HDAC2 Q92769 3/20 0.53
HDAC10 Q969S8 3/20 0.53
HDAC11 Q96DB2 3/20 0.53
HDAC8 Q9BY41 3/20 0.53
HDAC6 Q9UBN7 3/20 0.53
HDAC9 Q9UKV0 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7053721 0.80 DRD3 (0.72) DRD2DRD3DRD4FAAHHTR2A
SCHEMBL7051897 0.76 DRD2 (0.69) DRD2DRD3HTR2AHTR1AMEN1
SCHEMBL7114888 0.73 DRD2 (0.73) DRD2DRD3DRD4
SCHEMBL7054878 0.72 DRD2 (0.64) DRD2DRD3DRD4HTR2AHTR1A
SCHEMBL13808687 0.72 KMT2A (0.55) MEN1POLBRAB9AKMT2AHDAC3
SCHEMBL16403787 0.72 DRD3 (1.00) DRD2DRD3DRD4FAAHHTR2A
SCHEMBL9650947 0.72 DRD3 (0.75) DRD2DRD3DRD4HTR2AHTR1A
SCHEMBL5504452 0.70 DRD3 (1.00) DRD2DRD3DRD4HTR2AHTR1A
SCHEMBL8146978 0.70 KMT2A (0.82) MEN1POLBRAB9AKMT2AHDAC3
SCHEMBL5504457 0.70 DRD2 (0.70) DRD2DRD3DRD4HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028728-A1 4-(4-SUBSTITUTED PIPERAZINYL-1YL)-BUTYLCARBOXAMIDES AS D3 DOPAMINE SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed