SCHEMBL7057804

SCHEMBL7057804

COc1ccc(C(=O)NCCCCN2CCC(Nc3cc(F)ccc3F)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 9/20 0.63
DRD2 P14416 6/20 0.63
DRD4 P21917 2/20 0.55
HTR1A P08908 1/20 0.55
ADRA1D P25100 1/20 0.55
ADRA1A P35348 1/20 0.55
ADRA1B P35368 1/20 0.55
CCR3 P51677 2/20 0.54
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
CCR2 P41597 2/20 0.51
MAPT P10636 1/20 0.51
POLB P06746 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7057852 0.88 DRD3 (0.56) DRD3DRD2DRD4HTR1AADRA1D
SCHEMBL10724020 0.78 MAPT (0.75) DRD3DRD2NPC1RAB9AMAPT
SCHEMBL7055272 0.77 CCR3 (0.68) DRD3DRD2DRD4HTR1ACCR3
SCHEMBL20922354 0.75 POLB (0.61) DRD3DRD4CCR3NPC1RAB9A
SCHEMBL3124560 0.73 POLB (0.81) NPC1RAB9AMAPTPOLB
SCHEMBL229190 0.72 CYP2C9 (0.59) DRD3DRD2DRD4HTR1AADRA1D
Hydrochloric Acid SCHEMBL8820560 0.72 POLB (0.61) DRD4HTR1ACCR3MAPTPOLB
SCHEMBL9843330 0.72 HTR1A (0.88) DRD3DRD2DRD4HTR1AADRA1D
SCHEMBL9489987 0.72 NPC1 (1.00) NPC1RAB9APOLB
SCHEMBL11758269 0.72 NPC1 (1.00) NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003028725-A1 4-(1-PIPERIDINY)-BUTYLCARBOXAMIDE AS D3 DOPAMINE RECEPTOR SUBTYPE SELECTIVE LIGANDS Richter Gedeon Vegyészeti Gyár Rt. (HU) 2003-04-10 WO disclosed