SCHEMBL7058800

SCHEMBL7058800

O=C(CC1CC1c1ccccc1OC(F)(F)F)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.40
HTR2C P28335 8/20 0.40
HTR2B P41595 5/20 0.40
HTR2A P28223 2/20 0.40
DRD2 P14416 2/20 0.38
GAA P10253 1/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
RXRG P48443 1/20 0.36
FFAR1 O14842 1/20 0.36
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16586800 0.81 HTR2C (0.44) OPRM1HTR2CHTR2BHTR2AHCRTR1
SCHEMBL16586799 0.81 HTR2C (0.44) OPRM1HTR2CHTR2BHTR2AHCRTR1
SCHEMBL19262115 0.81 HTR2C (0.44) OPRM1HTR2CHTR2BHTR2AHCRTR1
SCHEMBL18016757 0.81 HTR2C (0.44) OPRM1HTR2CHTR2BHTR2AHCRTR1
SCHEMBL15254790 0.79 HTR2C (0.63) HTR2CHTR2BHTR2A
SCHEMBL16590861 0.79 HTR2C (0.49) HTR2CHTR2BHTR2AHCRTR1HCRTR2
SCHEMBL15254788 0.79 HTR2C (0.63) HTR2CHTR2BHTR2A
SCHEMBL18016882 0.75 HTR2C (0.49) OPRM1HTR2CHTR2BHTR2AHCRTR1
SCHEMBL17189661 0.74 DRD2 (0.44) OPRM1DRD2GAARXRARXRB
SCHEMBL2969140 0.74 DRD2 (0.44) OPRM1DRD2GAARXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490317-A1 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-12-29 EP disclosed
WO-2003082787-A1 GLUCOCORTICOID MIMETICS, METHODS OF MAKING THEM, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2003-10-09 WO disclosed