SCHEMBL7059210

SCHEMBL7059210

C=CCN(CC=C)S(=O)(=O)O

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
ESR1 P03372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11501152 0.97 KDM4E (0.36) KDM4EPOLBTDP1ALDH1A1MEN1
Benzene SCHEMBL10778436 0.93 RAB9A (0.40) KDM4EPOLBTDP1ALDH1A1MEN1
SCHEMBL11871750 0.82 RAB9A (0.47) KDM4EPOLBTDP1ALDH1A1MEN1
SCHEMBL973944 0.77 KDM4E (0.39) KDM4EPOLBTDP1ALDH1A1MEN1
SCHEMBL11031928 0.77 KDM4E (0.39) KDM4EPOLBTDP1ALDH1A1MEN1
SCHEMBL8652753 0.77 KDM4E (0.39) KDM4EPOLBTDP1ALDH1A1MEN1
SCHEMBL6431047 0.74 KDM4E (0.38) KDM4EPOLBTDP1ALDH1A1MEN1
Sulfuric Acid SCHEMBL28911116 0.74 ALDH1A1 (0.37) KDM4EPOLBTDP1ALDH1A1MEN1
SCHEMBL11668215 0.74
SCHEMBL7253370 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1075463-B1 CONVERSION OF A HYDROXY GROUP IN CERTAIN ALCOHOLS INTO A FLUOROSULFONATE ESTER OR A TRIFLUOROMETHYLSULFONATE ESTER LOEWENTHAL HANS JACOB EDGAR (IL) 2004-06-16 EP claimed
US-3939140-A Process for the preparation of a dyestuff consisting substantially of only unsymmetrical 1:2-chromium complex azo dyestuffs HOECHST AKTIENGESELLSCHAFT (DT) 1976-02-17 US claimed
US-11916195-B2 Electrolyte solution, electrochemical device, lithium ion secondary battery, and module DAIKIN INDUSTRIES, LTD. (JP) 2024-02-27 US disclosed
US-11916195-B2 Electrolyte solution, electrochemical device, lithium ion secondary battery, and module DAIKIN INDUSTRIES, LTD. (JP) 2024-02-27 US disclosed
US-20230387465-A1 COMPOUND, COMPOSITION, ELECTROCHEMICAL DEVICE, LITHIUM ION SECONDARY BATTERY AND MODULE DAIKIN INDUSTRIES, LTD. (JP) 2023-11-30 US disclosed
US-20230387465-A1 COMPOUND, COMPOSITION, ELECTROCHEMICAL DEVICE, LITHIUM ION SECONDARY BATTERY AND MODULE DAIKIN INDUSTRIES, LTD. (JP) 2023-11-30 US disclosed
US-20230145113-A1 ELECTROLYTIC SOLUTION, ELECTROCHEMICAL DEVICE, LITHIUM-ION SECONDARY BATTERY, MODULE AND COMPOUND DAIKIN INDUSTRIES, LTD. (JP) 2023-05-11 US disclosed
US-20230129817-A1 ELECTROLYTE SOLUTION, ELECTROCHEMICAL DEVICE, LITHIUM ION SECONDARY BATTERY AND MODULE DAIKIN INDUSTRIES, LTD. (JP) 2023-04-27 US disclosed
US-20230129817-A1 ELECTROLYTE SOLUTION, ELECTROCHEMICAL DEVICE, LITHIUM ION SECONDARY BATTERY AND MODULE DAIKIN INDUSTRIES, LTD. (JP) 2023-04-27 US disclosed
EP-4134994-A1 ELECTROLYTE SOLUTION, ELECTROCHEMICAL DEVICE, LITHIUM ION SECONDARY BATTERY AND MODULE Daikin Industries, Ltd. (JP) 2023-02-15 EP disclosed
EP-3933999-A1 ELECTROLYTIC SOLUTION, ELECTROCHEMICAL DEVICE, LITHIUM-ION SECONDARY BATTERY, MODULE AND COMPOUND DAIKIN INDUSTRIES, LTD. (JP) 2022-01-05 EP disclosed
EP-1075463-A1 CONVERSION OF A HYDROXY GROUP IN CERTAIN ALCOHOLS INTO A FLUOROSULFONATE ESTER OR A TRIFLUOROMETHYLSULFONATE ESTER Loewenthal, Hans Jacob Edgar (IL) 2001-02-14 EP disclosed
EP-0641355-B1 USE OF SULPHAMATE DERIVATIVES AS STEROID SULPHATASE INHIBITORS STERIX LTD (GB) 2000-07-19 EP disclosed
EP-0982032-A2 Use of a ring system compound comprising a sulphamic acid ester group for the manufacture of medicaments for the control of oestrogen production Sterix Limited (GB) 2000-03-01 EP disclosed
WO-1999055666-A1 CONVERSION OF A HYDROXY GROUP IN CERTAIN ALCOHOLS INTO A FLUOROSULFONATE ESTER OR A TRIFLUOROMETHYLSULFONATE ESTER LOEWENTHAL HANS JACOB EDGAR (IL) 1999-11-04 WO disclosed
EP-0928609-A2 Use of sulphamate derivatives as steroid sulphatase inhibitors IMPERIAL COLLEGE OF SCIENCE TECHNOLOGY AND MEDICINE (GB) 1999-07-14 EP disclosed
EP-0921130-A2 Steroid sulphatase inhibitors IMPERIAL COLLEGE OF SCIENCE, TECHNOLOGY & MEDICINE (GB) 1999-06-09 EP disclosed
US-5342444-A Pyrazolone dyes BAYER AKTIENGESELLSCHAFT (DE) 1994-08-30 US disclosed
US-4102924-A REACTING ACYLAMINO-ARYLS WITH HALO-ARYLS BAYER AKTIENGESELLSCHAFT (DE) 1978-07-25 US disclosed
US-3939140-A Process for the preparation of a dyestuff consisting substantially of only unsymmetrical 1:2-chromium complex azo dyestuffs HOECHST AKTIENGESELLSCHAFT (DT) 1976-02-17 US disclosed