Bromide

Bromide

SCHEMBL7060320

COc1cc2c(cc1OC)C(C)=[N+](Cc1ccccc1)CC2.[Br-]

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 10/20 0.48
KDM4E B2RXH2 1/20 0.48
GLA P06280 1/20 0.48
RCE1 Q9Y256 1/20 0.48
CHRNA7 P36544 1/20 0.43
DNMT1 P26358 1/20 0.42
KDM1A O60341 1/20 0.42
COL1A1 P02452 2/20 0.41
NR1H4 Q96RI1 1/20 0.41
BCHE P06276 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14131507 0.99 ACHE (0.49) ACHEKDM4EGLARCE1CHRNA7
SCHEMBL4764328 0.86 ACHE (0.51) ACHEKDM4EDNMT1KDM1ACOL1A1
Hydrochloric Acid SCHEMBL4110961 0.85 ACHE (0.50) ACHEKDM4EDNMT1KDM1ACOL1A1
SCHEMBL4771879 0.82 ACHE (0.46) ACHEKDM4EGLARCE1DNMT1
SCHEMBL4762866 0.82 MAPT (0.43) ACHEKDM4EDNMT1KDM1ACOL1A1
SCHEMBL4837359 0.82 COL1A1 (0.48) ACHEDNMT1KDM1ACOL1A1BCHE
Bromide SCHEMBL10708277 0.82 ACHE (0.42) ACHEKDM4EGLARCE1CHRNA7
Hydrochloric Acid SCHEMBL4109381 0.81 ACHE (0.45) ACHEKDM4EGLARCE1DNMT1
Hydrochloric Acid SCHEMBL4097637 0.81 MAPT (0.42) ACHEKDM4EDNMT1KDM1ACOL1A1
Hydrochloric Acid SCHEMBL4098744 0.81 COL1A1 (0.47) ACHEDNMT1KDM1ACOL1A1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117627-B1 TRANSFER HYDROGENATION PROCESS AVECIA LTD (GB) 2003-05-28 EP disclosed
US-6509467-B1 Of iminium salts using transition metal complex catalyst AVECIA LIMITED (GB) 2003-01-21 US disclosed
EP-1117627-A1 TRANSFER HYDROGENATION PROCESS Avecia Limited (GB) 2001-07-25 EP disclosed
WO-2000018708-A1 TRANSFER HYDROGENATION PROCESS AVECIA LIMITED (GB) 2000-04-06 WO disclosed