SCHEMBL7065148

SCHEMBL7065148

CCOC(=O)c1cn(C[C@H]2CC[C@H]3C(CC)N[C@H](C(=O)O)C[C@H]3C2)cn1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.33
NOTUM Q6P988 1/20 0.32
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7065326 0.99 USP30 (0.33) USP30NOTUM
SCHEMBL7068740 0.96 USP30 (0.33) USP30NOTUM
SCHEMBL7070985 0.83 TP53 (0.32) LMNA
Hydrochloric Acid SCHEMBL7066446 0.83 TP53 (0.31) LMNA
Hydrochloric Acid SCHEMBL7071085 0.81 GRIK1 (0.45)
SCHEMBL7064873 0.81 TP53 (0.30)
Hydrochloric Acid SCHEMBL7068329 0.80 TP53 (0.30)
Hydrochloric Acid SCHEMBL7066458 0.79 GABRA1 (0.36) LMNA
SCHEMBL7066186 0.77 USP30 (0.33) USP30NOTUMLMNA
SCHEMBL7065145 0.77 USP30 (0.36) USP30NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6579886-B2 Ionotropic glutamate receptors; 6-((4-carboxylic acid-1H-imidazol-1-yl)methyl)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3 -carboxylic acid ELI LILLY AND COMPANY 2003-06-17 US claimed
US-20030055081-A1 Selective iglur5 receptor antagonists ELI LILLY AND COMPANY 2003-03-20 US claimed
US-6579886-B2 Ionotropic glutamate receptors; 6-((4-carboxylic acid-1H-imidazol-1-yl)methyl)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3 -carboxylic acid ELI LILLY AND COMPANY 2003-06-17 US disclosed
US-20030055081-A1 Selective iglur5 receptor antagonists ELI LILLY AND COMPANY 2003-03-20 US disclosed
EP-1257545-A1 SELECTIVE iGLUR 5? RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2002-11-20 EP disclosed
WO-2001046173-A1 SELECTIVE iGLUR5 RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2001-06-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030055081-A1 Selective iglur5 receptor antagonists GRM5, GRIK5, GPR35 USP30 2572/4885NOTUM 1912/4885LMNA 3014/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.