SCHEMBL7068322

SCHEMBL7068322

COc1cc(OC2CCN(C)CC2)c2c(Nc3cccc4ccoc34)c(C#N)cnc2c1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SRC P12931 13/20 0.49
KDR P35968 3/20 0.49
ABL1 P00519 7/20 0.48
ABL2 P42684 7/20 0.48
EGFR P00533 5/20 0.45
ERBB2 P04626 2/20 0.45
FLT1 P17948 1/20 0.44
RAF1 P04049 1/20 0.44
MAP2K1 Q02750 1/20 0.44
IKBKE Q14164 1/20 0.40
TBK1 Q9UHD2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7067904 0.99 SRC (0.48) SRCKDRABL1ABL2EGFR
SCHEMBL7065293 0.89 SRC (0.46) SRCABL1ABL2EGFRERBB2
Hydrochloric Acid SCHEMBL7070735 0.88 SRC (0.45) SRCABL1ABL2EGFRERBB2
SCHEMBL7068505 0.87 SRC (0.50) SRCKDRABL1ABL2EGFR
SCHEMBL7068176 0.83 SRC (0.52) SRCKDRABL1ABL2EGFR
Hydrochloric Acid SCHEMBL7066964 0.83 SRC (0.70) SRCKDRABL1ABL2EGFR
SCHEMBL7065518 0.83 SRC (0.49) SRCKDRABL1EGFRRAF1
Hydrochloric Acid SCHEMBL7068675 0.82 SRC (0.49) SRCKDRABL1EGFRRAF1
Hydrochloric Acid SCHEMBL3279304 0.82 SRC (0.69) SRCKDREGFRERBB2
SCHEMBL5471839 0.78 SRC (0.51) SRCKDRABL1ABL2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003047583-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING BENZOFURANYL SUBSTITUTED 3-CYANOQUINOLINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF SOLID TUMOURS ASTRAZENECA AB (SE) 2003-06-12 WO disclosed
WO-2003048159-A1 QUINOLINE DERIVATIVES ASTRAZENECA AB (SE) 2003-06-12 WO disclosed