SCHEMBL7071124

SCHEMBL7071124

CC(C)C(NC(=O)OC(C)(C)C)C(=O)c1nnc(C(C)(C)c2ccccc2)o1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ELANE P08246 13/20 0.54
TRPA1 O75762 2/20 0.46
CTSK P43235 3/20 0.43
CTSS P25774 2/20 0.43
MAPT P10636 1/20 0.41
ATM Q13315 1/20 0.41
CTSL P07711 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7068029 0.84 ELANE (0.49) ELANETRPA1CTSKCTSS
SCHEMBL7007704 0.77 ELANE (0.55) ELANE
Hydrochloric Acid SCHEMBL7075284 0.76 ELANE (0.48) ELANEMAPT
SCHEMBL7199762 0.75 ELANE (0.71) ELANE
SCHEMBL7438422 0.74 TRPA1 (0.57) TRPA1CTSKCTSSATMCTSL
SCHEMBL8283003 0.74 TRPA1 (0.57) TRPA1CTSKCTSSATMCTSL
SCHEMBL7956686 0.74 ELANE (0.48) ELANEMAPT
SCHEMBL7158995 0.73 ELANE (0.89) ELANE
SCHEMBL27158525 0.73 PTPN1 (0.46) ELANEMAPT
SCHEMBL30522758 0.71 TRPA1 (0.46) TRPA1CTSKCTSSMAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030153758-A1 1,3,4-Oxadiazole derivatives and process for producing the same ONO PHARMACEUTICAL CO., LTD. 2003-08-14 US claimed
US-6534658-B1 Intermediates for producing pharmaceuticals ONO PHARMACEUTICAL CO., LTD. (JP) 2003-03-18 US claimed
EP-1162199-A1 1,3,4-OXADIAZOLE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME ONO PHARMACEUTICAL CO., LTD. (JP) 2001-12-12 EP claimed
US-20030153758-A1 1,3,4-Oxadiazole derivatives and process for producing the same ONO PHARMACEUTICAL CO., LTD. 2003-08-14 US disclosed
US-6534658-B1 Intermediates for producing pharmaceuticals ONO PHARMACEUTICAL CO., LTD. (JP) 2003-03-18 US disclosed
EP-1162199-A1 1,3,4-OXADIAZOLE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME ONO PHARMACEUTICAL CO., LTD. (JP) 2001-12-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030153758-A1 1,3,4-Oxadiazole derivatives and process for producing the same OXA1L, CYP1B1, OXER1 ELANE 4189/4885TRPA1 2697/4885CTSK 3506/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.