SCHEMBL7072061

SCHEMBL7072061

O=C(O)Oc1cc2c(-c3cccnc3)cccc2n1Cc1ccc(Cl)c(Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 15/20 0.58
PTGDR2 Q9Y5Y4 1/20 0.42
DHPS P49366 1/20 0.41
MAPK14 Q16539 1/20 0.41
PTGES2 Q9H7Z7 1/20 0.41
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7072260 0.85 CCR2 (0.59) CCR2ALDH1A1LMNACYP1A2CYP3A4
SCHEMBL6300535 0.85 CCR2 (0.80) CCR2
SCHEMBL7076325 0.85 CCR2 (0.56) CCR2ALDH1A1LMNACYP1A2CYP3A4
SCHEMBL7072428 0.83 CCR2 (0.53) CCR2PTGDR2MAPK14ALDH1A1LMNA
SCHEMBL7076059 0.82 CCR2 (0.68) CCR2ALDH1A1LMNACYP1A2CYP3A4
SCHEMBL6307932 0.80 CCR2 (0.61) CCR2PTGDR2MAPK14LMNAMAPT
SCHEMBL7077386 0.80 CCR2 (0.56) CCR2ALDH1A1LMNACYP1A2CYP3A4
SCHEMBL7072264 0.80 CCR2 (0.52) CCR2ALDH1A1LMNACYP1A2CYP3A4
SCHEMBL7080358 0.79 CCR2 (0.70) CCR2ALDH1A1LMNACYP1A2CYP3A4
SCHEMBL7077403 0.79 CCR2 (0.70) CCR2ALDH1A1LMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003504-B1 INDOLE DERIVATIVES AND THEIR USE AS MCP-1 ANTAGONISTS ASTRAZENECA AB (SE) 2003-07-02 EP claimed