SCHEMBL7072933

SCHEMBL7072933

O=CC(Br)c1c(Br)cc(Br)cc1Br

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.39
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
GABRA1 P14867 1/20 0.31
GABRB1 P18505 1/20 0.31
GABRA2 P47869 1/20 0.31
GABRB2 P47870 1/20 0.31
PTPN1 P18031 1/20 0.31
AKR1C4 P17516 1/20 0.30
AKR1C3 P42330 1/20 0.30
AKR1C2 P52895 1/20 0.30
AKR1C1 Q04828 1/20 0.30
HSP90AA1 P07900 1/20 0.30
TLR9 Q9NR96 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23754492 0.77 DGAT1 (0.31)
SCHEMBL2572781 0.76 CYP2A6 (0.33)
SCHEMBL861863 0.74 GABRA1 (0.47) GABRA1GABRB1
SCHEMBL4091711 0.68 TDP1 (0.45) ERN1CYP3A4TSHRTDP1GABRA1
SCHEMBL18243263 0.67 CYP3A4 (0.39) ERN1CYP3A4TSHRTDP1GABRA1
SCHEMBL10832001 0.67 CYP3A4 (0.39) CYP3A4TSHRTDP1GABRA1GABRB1
SCHEMBL3979239 0.67 ERN1 (0.39) ERN1CYP3A4TSHRTDP1PTPN1
SCHEMBL9772766 0.66
SCHEMBL20551266 0.65 ERN1 (0.38) ERN1
SCHEMBL22833975 0.65 ERN1 (0.32) ERN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003055479-A1 COMPOUNDS AND THEIR THERAPEUTIC USE RELATED TO THE PHOSPHORYLATING ACTIVITY OF THE ENZYME GSK-3 CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS (ES) 2003-07-10 WO disclosed