SCHEMBL7073157

SCHEMBL7073157

COC(=O)Cc1cc(C)c(Oc2ccc(O)c(C(C)C)c2)c(Cl)c1

nearest known ligand 0.69

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
THRA P10827 12/20 0.69
THRB P10828 12/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4558899 0.89 THRA (0.87) THRATHRB
SCHEMBL7073438 0.88 THRA (0.67) THRATHRB
SCHEMBL7643749 0.82 THRB (0.58) THRATHRB
SCHEMBL5281917 0.82 THRA (0.78) THRATHRB
SCHEMBL282382 0.82 THRA (1.00) THRATHRB
SCHEMBL29373235 0.82 THRA (1.00) THRATHRB
SCHEMBL19057792 0.82 THRB (0.82) THRATHRB
SCHEMBL7073126 0.80 THRA (0.76) THRATHRB
SCHEMBL282637 0.80 THRB (0.54) THRATHRB
SCHEMBL4964368 0.77 THRB (0.63) THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000008-B1 NOVEL THYROID RECEPTOR LIGANDS AND METHOD KAROBIO AB (SE) 2003-06-25 EP disclosed
US-6465687-B1 SUBSTITUTED 4-HYDROXY-3-ALKYL- OR CYCLOALKYL-PHENOXYBENZENE COMPOUNDS SUCH AS 3,5-DIBROMO-4-(4-HYDROXY-3-ISOPROPYLPHENOXY)BENZOIC ACID, EXPRESSION INHIBITION OF A T3 REGULATED GENE KARO BIO AB (SE) 2002-10-15 US disclosed
EP-1000008-A1 NOVEL THYROID RECEPTOR LIGANDS AND METHOD KARO BIO AB (SE) 2000-05-17 EP disclosed
WO-1999000353-A1 NOVEL THYROID RECEPTOR LIGANDS AND METHOD KARO BIO AB (SE) 1999-01-07 WO disclosed