SCHEMBL7073345

SCHEMBL7073345

CC(C)(C)OC(=O)N1CCc2[nH]c3ccccc3c2CC1.CC(C)(C)OC(=O)N1CCc2c(n(CCS(=O)(=O)c3ccccc3)c3ccccc23)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
TRPV1 Q8NER1 5/20 0.42
FAAH O00519 2/20 0.42
HTR6 P50406 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
BAZ2B Q9UIF8 1/20 0.41
GPX4 P36969 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
CNR2 P34972 1/20 0.38
F12 P00748 1/20 0.38
SSTR3 P32745 1/20 0.37
KMT2A Q03164 1/20 0.37
ENPP2 Q13822 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6475467 0.92 HDAC1 (0.51) HDAC1HDAC6HTR6LMNACHRM2
SCHEMBL6786012 0.84 HDAC1 (0.47) HDAC1HDAC6TRPV1FAAHLMNA
SCHEMBL7466922 0.83 HDAC1 (0.46) HDAC1HDAC6TRPV1FAAHLMNA
SCHEMBL6474214 0.80 LMNA (0.60) TRPV1FAAHLMNAMAPTBAZ2B
SCHEMBL6474858 0.79 HDAC1 (0.51) HDAC1HDAC6HTR6CHRM2CHRM4
SCHEMBL6480968 0.79 KDM4E (0.49) HTR6PTGDR2KMT2AENPP2
SCHEMBL6474153 0.78 KDM4E (0.61) HDAC1HDAC6BAZ2BCHRM2CHRM4
SCHEMBL6475292 0.78 HDAC1 (0.56) HDAC1HDAC6CHRM2CHRM4CHRM1
SCHEMBL7069900 0.77 KDM4E (0.60) HDAC1HDAC6BAZ2BCHRM2CHRM4
SCHEMBL6475536 0.77 HDAC1 (0.55) HDAC1HDAC6CHRM2CHRM4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1319004-A2 SUBSTITUTED AZEPINO[4,5-B]INDOLE DERIVATIVES PHARMACIA & UPJOHN COMPANY (US) 2003-06-18 EP disclosed
WO-2002024701-A2 SUBSTITUTED AZEPINO[4,5B)INDOLE DERIVATIVES PHARMACIA & UPJOHN COMPANY (US) 2002-03-28 WO disclosed