SCHEMBL7074302

SCHEMBL7074302

N=C(N)c1ccc(C(=O)N2CCN(S(=O)(=O)c3cccc(Cl)c3Cl)CC2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 2/20 0.53
TSHR P16473 1/20 0.52
KMT2A Q03164 4/20 0.48
LMNA P02545 3/20 0.48
MMP2 P08253 1/20 0.47
MMP13 P45452 1/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CHRM1 P11229 1/20 0.46
POLB P06746 1/20 0.46
MEN1 O00255 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL27550418 0.96 F10 (0.49) F10TSHRKMT2ALMNAMMP2
SCHEMBL7071342 0.83 CNR1 (0.57) F10TSHRKMT2ALMNAMMP2
SCHEMBL7074838 0.82 F10 (0.54) F10TSHRKMT2ALMNAMMP2
SCHEMBL7074161 0.81 KMT2A (0.58) F10TSHRKMT2AALDH1A1MAPT
SCHEMBL7072134 0.80 F10 (0.63) F10KMT2ALMNAALDH1A1GAA
Acetic Acid SCHEMBL27538655 0.80 CNR1 (0.53) F10TSHRKMT2ALMNAMMP2
SCHEMBL7071636 0.79 F10 (0.53) F10KMT2ALMNAALDH1A1POLB
Acetic Acid SCHEMBL27550443 0.79 LMNA (0.52) F10TSHRKMT2ALMNAMMP2
SCHEMBL7077553 0.79 F10 (0.65) F10KMT2ALMNAMAPTCA12
SCHEMBL7074220 0.79 LMNA (0.71) F10KMT2ALMNAALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-B1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 2003-06-25 EP disclosed
US-6492368-B1 Benzamidine derivatives as factor XA inhibitors MERCK PATENT GMBH (DE) 2002-12-10 US disclosed