SCHEMBL7076834

SCHEMBL7076834

O=C(O)c1cccc(Nc2ccc3ccccc3c2)c1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.65
CYP3A4 P08684 1/20 0.65
HPGD P15428 1/20 0.65
HSD17B10 Q99714 1/20 0.65
RHOA P61586 1/20 0.64
MRGPRX4 Q96LA9 1/20 0.62
AKR1C3 P42330 5/20 0.61
AKR1C2 P52895 3/20 0.59
CSNK2A1 P68400 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.57
CDC25B P30305 4/20 0.57
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
MAPT P10636 1/20 0.56
SIRT2 Q8IXJ6 1/20 0.55
SIRT1 Q96EB6 1/20 0.55
SIRT3 Q9NTG7 1/20 0.55
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7524753 0.86 ALDH1A1 (0.69) ALDH1A1CYP3A4HPGDHSD17B10MRGPRX4
3-Phenylamino Benzoic Acid SCHEMBL4345076 0.86 RHOA (0.77) ALDH1A1HPGDHSD17B10RHOAAKR1C3
Diphenylamine SCHEMBL28427475 0.80 ALDH1A1 (0.64) ALDH1A1CYP3A4HPGDHSD17B10RHOA
SCHEMBL22651908 0.80 ALDH1A1 (0.91) ALDH1A1CYP3A4HPGDHSD17B10L3MBTL1
SCHEMBL9486049 0.80 ALDH1A1 (0.91) ALDH1A1CYP3A4HPGDHSD17B10L3MBTL1
SCHEMBL11466814 0.80 ALDH1A1 (1.00) ALDH1A1CYP3A4HPGDHSD17B10L3MBTL1
SCHEMBL29354421 0.80 ALDH1A1 (1.00) ALDH1A1CYP3A4HPGDHSD17B10L3MBTL1
SCHEMBL7928040 0.80 ALDH1A1 (0.83) ALDH1A1CYP3A4HPGDHSD17B10L3MBTL1
SCHEMBL38433 0.80 ALDH1A1 (1.00) ALDH1A1CYP3A4HPGDHSD17B10L3MBTL1
Benzene SCHEMBL28342167 0.80 ALDH1A1 (1.00) ALDH1A1CYP3A4HPGDHSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944582-B1 KETOBENZAMIDES AS CALPAIN INHIBITORS ABBOTT GMBH & CO KG (DE) 2003-07-02 EP disclosed
EP-0944582-A1 KETOBENZAMIDES AS CALPAIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-09-29 EP disclosed
EP-0944584-A1 BENZAMIDOALDEHYDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1999-09-29 EP disclosed
WO-1998025883-A1 KETOBENZAMIDES AS CALPAIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-06-18 WO disclosed
WO-1998023581-A1 BENZAMIDOALDEHYDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-06-04 WO disclosed