SCHEMBL7077929

SCHEMBL7077929

CC(C)NC1=NS(=O)(=O)c2scc(Cl)c2N1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 2/20 0.31
CXCR1 P25024 1/20 0.30
NT5E P21589 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8475613 0.85
SCHEMBL8475723 0.84
SCHEMBL7078037 0.83
SCHEMBL8474127 0.79 PDE4B (0.34)
SCHEMBL8473769 0.78 HPGD (0.36) CXCR2
SCHEMBL7076103 0.77
SCHEMBL7073682 0.75 NT5E (0.30) NT5E
SCHEMBL7079890 0.75 NT5E (0.30) NT5E
SCHEMBL8474564 0.74
SCHEMBL8476651 0.74 NT5E (0.30) NT5E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030235583-A1 Combined use of a modulator of CD3 and a beta cell resting compound NOVO NORDISK A/S (DK) 2003-12-25 US claimed
US-20030125323-A1 Use of selective potassium channel openers NOVO NORDISK A/S (DK) 2003-07-03 US claimed
US-20030109519-A1 Use of selective potassium channel openers NOVO NORDISK (DK) 2003-06-12 US claimed
US-20020035106-A1 Use of potassium channel agonists for reducing fat food consumption NOVO NORDISK A/S (DK) 2002-03-21 US claimed
US-20020028808-A1 Use of potassium channel agonists for the treatment of cancer NOVO NORDISK A/S (DK) 2002-03-07 US claimed
US-6225310-B1 Fused 1,2,4-thiadiazine derivatives, their preparation and use NOVO NORDISK A/S (DK) 2001-05-01 US claimed
CN-1264384-A Fused 1,2,4-thiadiazine derivatives, their preparation method and use NOVO NORDISK AS (DK) 2000-08-23 CN claimed
US-20030235583-A1 Combined use of a modulator of CD3 and a beta cell resting compound NOVO NORDISK A/S (DK) 2003-12-25 US disclosed
US-20030125323-A1 Use of selective potassium channel openers NOVO NORDISK A/S (DK) 2003-07-03 US disclosed
US-20030109519-A1 Use of selective potassium channel openers NOVO NORDISK (DK) 2003-06-12 US disclosed
WO-2003045955-A1 USE OF SELECTIVE POTASSIUM CHANNEL OPENERS NOVO NORDISK A/S (DK) 2003-06-05 WO disclosed
US-20020035106-A1 Use of potassium channel agonists for reducing fat food consumption NOVO NORDISK A/S (DK) 2002-03-21 US disclosed
US-20020028808-A1 Use of potassium channel agonists for the treatment of cancer NOVO NORDISK A/S (DK) 2002-03-07 US disclosed
US-6225310-B1 Fused 1,2,4-thiadiazine derivatives, their preparation and use NOVO NORDISK A/S (DK) 2001-05-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030125323-A1 Use of selective potassium channel openers KCNJ11, KCNJ1, KCNJ2 CXCR2 4185/4885CXCR1 3080/4885NT5E 2763/4885
US-20030109519-A1 Use of selective potassium channel openers KCNJ11, KCNJ2, KCNJ1 CXCR2 4038/4885CXCR1 2805/4885NT5E 1982/4885
US-20020028808-A1 Use of potassium channel agonists for the treatment of cancer KCNN3, KCNN1, KCNN2 CXCR2 3575/4885CXCR1 3717/4885NT5E 1702/4885
US-20030235583-A1 Combined use of a modulator of CD3 and a beta cell resting compound CD69, IAPP, CD4 CXCR2 2526/4885CXCR1 608/4885NT5E 1205/4885
US-20020035106-A1 Use of potassium channel agonists for reducing fat food consumption KCNN3, KCNN2, KCNN1 CXCR2 3688/4885CXCR1 3971/4885NT5E 1624/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.