SCHEMBL7078434

SCHEMBL7078434

CC(C)(C)OC(=O)c1cc(Br)cc(C(=O)O)c1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.42
KDM4E B2RXH2 3/20 0.42
GLA P06280 1/20 0.42
AKR1C3 P42330 2/20 0.40
AKR1C2 P52895 2/20 0.40
AKR1C1 Q04828 2/20 0.40
AKR1C4 P17516 1/20 0.40
LCK P06239 1/20 0.34
FYN P06241 1/20 0.34
GRM6 O15303 1/20 0.34
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
CA14 Q9ULX7 2/20 0.33
CA3 P07451 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6232764 0.85 SLC7A5 (0.40) HSD17B10KDM4EGRM6CA12CA1
SCHEMBL1767847 0.85 KDM4E (0.40) HSD17B10KDM4EGRM6CA12CA1
SCHEMBL7074918 0.85 KDM4E (0.56) KDM4EGRM6CA12CA1CA2
SCHEMBL7075526 0.84 KEAP1 (0.42) HSD17B10KDM4EGRM6CA12CA1
SCHEMBL7324883 0.84 LCK (0.39) HSD17B10KDM4ELCKGRM6CA12
SCHEMBL7071957 0.84 CYP3A4 (0.46) HSD17B10KDM4EGLAAKR1C3AKR1C2
SCHEMBL28992396 0.81 KDM4E (0.44) HSD17B10KDM4EGLAAKR1C3AKR1C2
SCHEMBL15920614 0.79 KDM4E (0.47) HSD17B10KDM4EGLAMYCNR4A1
SCHEMBL4628585 0.79 KDM4E (0.47) HSD17B10KDM4EGLAMYCNR4A1
SCHEMBL27996077 0.78 CA12 (0.42) HSD17B10KDM4EGLAGRM6CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003052053-A2 NUCLEOSIDE LIBRARIES AND COMPOUNDS BY MCC COMBINATORIAL STRATEGIES ON SOLID SUPPORT RIBAPHARM INC. (US) 2003-06-26 WO disclosed