SCHEMBL7078503

SCHEMBL7078503

CC(C)(C)[Si](C)(C)OCc1cn(-c2ccc(N3C[C@H](COc4ccon4)OC3=O)cc2F)cn1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 10/20 0.39
MAOB P27338 8/20 0.37
CALML3 P27482 2/20 0.36
LMNA P02545 1/20 0.36
PTGS1 P23219 1/20 0.36
SDHA P31040 1/20 0.36
GRM2 Q14416 4/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084731 1.00 MAOA (0.39) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL7077047 0.87 MAOA (0.42) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL7077051 0.87 MAOA (0.42) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL7081049 0.86 MAOA (0.46) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL3753819 0.86 MAOA (0.41) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL4012835 0.86 MAOA (0.41) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL3757473 0.86 CALML3 (0.48) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL5833572 0.86 CALML3 (0.48) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL7081053 0.86 MAOA (0.46) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL3755980 0.85 MAOB (0.43) MAOAMAOBCALML3LMNAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6617339-B1 5-Isoxazolyloxymethyl-3-((dihydroxypropanoyl)-4-tetrahydropyri dyl-3,5- difluorophenyl)oxazolidinone, or the phosphated derivative or its disodium salt; antibiotic with useful activity against Grampositive pathogens SYNGENTA LIMITED (GB) 2003-09-09 US disclosed
US-20030144263-A1 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them SYNGENTA LIMITED (GB) 2003-07-31 US disclosed
EP-1082323-A2 OXAZOLIDINONE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AstraZeneca UK Limited (GB) 2001-03-14 EP disclosed
WO-1999064417-A2 OXAZOLIDINONE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ASTRAZENECA AB (SE) 1999-12-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030144263-A1 Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them CYP3A5, CYP2D6, OXA1L MAOA 1654/4885MAOB 1178/4885CALML3 4622/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.