SCHEMBL7078784

SCHEMBL7078784

Nc1cccc(C(=O)NCCN2CC3CC(c4ccc(Cl)cc4)C3C2)c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 7/20 0.45
DRD4 P21917 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
DRD2 P14416 1/20 0.43
PMP22 Q01453 1/20 0.43
EPHX2 P34913 1/20 0.43
KCNH2 Q12809 4/20 0.43
ALDH1A1 P00352 2/20 0.42
POLB P06746 1/20 0.42
HTR1A P08908 2/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
CD274 Q9NZQ7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7071623 0.88 ALDH1A1 (0.51) MCHR1CYP1A2DRD2PMP22EPHX2
SCHEMBL7774081 0.83 ALDH1A1 (0.50) MCHR1DRD4CYP1A2CYP3A4CYP2D6
SCHEMBL7075387 0.82 ALDH1A1 (0.44) CYP1A2CYP3A4CYP2D6KCNH2ALDH1A1
SCHEMBL7778723 0.81 ALDH1A1 (0.48) DRD4CYP1A2CYP3A4CYP2D6MAPT
SCHEMBL7817609 0.80 HTR1A (0.46) MCHR1DRD4CYP1A2CYP2D6DRD2
SCHEMBL8989768 0.80 ALDH1A1 (0.49) DRD2EPHX2KCNH2ALDH1A1HTR1A
SCHEMBL7778722 0.80 KDM1A (0.50) CD274
Cyclohexane SCHEMBL7076604 0.79 ALDH1A1 (0.43) KCNH2ALDH1A1HTR1AMAOAMAOB
Cyclopentane SCHEMBL7071122 0.79 ALDH1A1 (0.43) KCNH2ALDH1A1HTR1AMAOAMAOB
SCHEMBL8989722 0.78 DRD4 (0.55) MCHR1DRD4CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0740658-B1 N-SUBSTITUTED AZABICYCLOHEPTANE DERIVATIVES USED, FOR EXAMPLE, AS NEUROLEPTICS ABBOTT GMBH & CO KG (DE) 2003-07-02 EP disclosed
US-5616705-A N-substituted azabicycloheptane derivatives, their preparation and use BASF AKTIENGESELLSCHAFT (DE) 1997-04-01 US disclosed
EP-0740658-A1 N-SUBSTITUTED AZABICYCLOHEPTANE DERIVATIVES USED, FOR EXAMPLE, AS NEUROLEPTICS BASF AKTIENGESELLSCHAFT (DE) 1996-11-06 EP disclosed
WO-1995015312-A1 N-SUBSTITUTED AZABICYCLOHEPTANE DERIVATIVES USED, FOR EXAMPLE, AS NEUROLEPTICS BASF AKTIENGESELLSCHAFT (DE) 1995-06-08 WO disclosed