SCHEMBL7079844

SCHEMBL7079844

COc1ccccc1COC1CN(OC(=O)OC(C)(C)C)CCC1c1ccc(OCc2ccc3ccccc3c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
REN P00797 18/20 0.51
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM1A O60341 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7074891 0.91 REN (0.48) REN
SCHEMBL7085119 0.89 REN (0.58) REN
SCHEMBL7077892 0.87 REN (0.42) RENKDM1AMAOAMAOB
SCHEMBL6953596 0.86 REN (0.55) REN
SCHEMBL7076933 0.86 REN (0.43) RENMEN1KMT2A
SCHEMBL7080924 0.86 REN (0.54) REN
SCHEMBL7075237 0.86 REN (0.56) REN
SCHEMBL7078693 0.86 REN (0.49) REN
SCHEMBL7078656 0.86 REN (0.54) REN
SCHEMBL7083053 0.86 REN (0.47) REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863875-B1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY HOFFMANN LA ROCHE (CH) 2003-06-04 EP disclosed
EP-0863875-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1998-09-16 EP disclosed
WO-1997009311-A1 NEW 4-(OXYALKOXYPHENYL)-3-OXY-PIPERIDINES FOR TREATING HEART AND KIDNEY INSUFFICIENCY F. HOFFMANN-LA ROCHE AG (CH) 1997-03-13 WO disclosed