SCHEMBL7080045

SCHEMBL7080045

CC(C)c1nc(CCO)n(CCc2ccccc2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.37
KMT2A Q03164 5/20 0.37
LMNA P02545 3/20 0.37
POLB P06746 2/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 2/20 0.36
CASR P41180 2/20 0.34
ALDH1A1 P00352 5/20 0.34
CASP1 P29466 4/20 0.34
HIF1A Q16665 4/20 0.34
HSD17B10 Q99714 4/20 0.34
CYP3A4 P08684 4/20 0.34
CASP7 P55210 3/20 0.34
CYP2C9 P11712 3/20 0.34
CYP2C19 P33261 3/20 0.34
CYP1A2 P05177 2/20 0.34
USP2 O75604 2/20 0.34
GLA P06280 1/20 0.34
HBB P68871 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974514 0.94 MEN1 (0.35) MEN1KMT2ALMNAPOLBGAA
SCHEMBL6973318 0.94 MAPK14 (0.38) MEN1KMT2ALMNAPOLBALDH1A1
SCHEMBL6961236 0.93 POLB (0.44) MEN1KMT2ALMNAPOLBGAA
SCHEMBL6964205 0.91 HRH1 (0.32) MEN1KMT2A
SCHEMBL6974234 0.91 TDP1 (0.36) LMNAALDH1A1HSD17B10SMN1; SMN2HTT
SCHEMBL6969724 0.89 MAPK14 (0.37) MEN1KMT2APOLBALDH1A1CYP2C9
SCHEMBL6968588 0.88 MEN1 (0.37) MEN1KMT2ALMNAPOLBGAA
SCHEMBL6965421 0.87 POLB (0.38) MEN1KMT2ALMNAPOLBALDH1A1
SCHEMBL6963837 0.86 MEN1 (0.37) MEN1KMT2AMAPTALDH1A1HPGD
SCHEMBL6966608 0.85 MAPK14 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed