SCHEMBL7080073

SCHEMBL7080073

C=CCc1cc([N+](=O)[O-])ccc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRC P08575 1/20 0.41
S100A4 P26447 1/20 0.41
ALDH1A1 P00352 4/20 0.40
TDP1 Q9NUW8 4/20 0.40
CYP3A4 P08684 1/20 0.40
POLB P06746 3/20 0.39
MAPT P10636 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 2/20 0.38
TSHR P16473 2/20 0.38
LMNA P02545 1/20 0.38
CA2 P00918 2/20 0.38
CA5A P35218 2/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA3 P07451 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA7 P43166 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5748776 0.85 PTPRC (0.42) PTPRCS100A4ALDH1A1TDP1CYP3A4
SCHEMBL9683795 0.81 TDP1 (0.50) ALDH1A1TDP1CYP3A4POLBMAPT
SCHEMBL27401907 0.80 HSD17B10 (0.55) ALDH1A1TDP1MAPTMEN1KMT2A
SCHEMBL2552755 0.80 ALDH1A1 (0.55) ALDH1A1TDP1CYP3A4POLBMAPT
SCHEMBL4980531 0.80 POLB (0.61) ALDH1A1TDP1POLBMAPTMEN1
SCHEMBL532452 0.79 PTPRC (0.46) PTPRCS100A4ALDH1A1TDP1CYP3A4
SCHEMBL13043154 0.79 POLB (0.53) PTPRCS100A4ALDH1A1TDP1CYP3A4
SCHEMBL30279963 0.79 PTPRC (0.46) PTPRCS100A4ALDH1A1TDP1CYP3A4
SCHEMBL4301056 0.79 MEN1 (0.45) ALDH1A1TDP1POLBMAPTMEN1
SCHEMBL11097917 0.79 TSHR (0.44) PTPRCS100A4ALDH1A1TDP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1013636-B1 Preparation of allylic aromatic compounds AMERSHAM HEALTH AS (NO) 2003-07-09 EP disclosed
US-6284894-B1 AROMATIC AMINE IS REACTED FIRST WITH A NITRITE AND THEN WITH AN ALLYLIC OLEFIN HAVING AN ELIMINATABLE TERMINAL SUBSTITUENT. NYCOMED IMAGING AS (NO) 2001-09-04 US disclosed
EP-1013636-A1 Preparation of allylic aromatic compounds NYCOMED IMAGING AS (NO) 2000-06-28 EP disclosed