SCHEMBL7081248

SCHEMBL7081248

CO/N=C1\C[C@@H](C(=O)NC[C@@H](O)c2ccccc2)N(C(=O)c2ccc(-c3ccccc3OC)cc2)C1

nearest known ligand 0.85

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OXTR P30559 5/20 0.85
AVPR1A P37288 3/20 0.85
FFAR2 O15552 13/20 0.45
ROCK2 O75116 2/20 0.41
ROCK1 Q13464 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7089044 1.00 OXTR (0.85) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4939000 1.00 OXTR (0.85) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL7088046 0.94 OXTR (0.76) OXTRAVPR1AFFAR2
SCHEMBL5743780 0.92 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4936354 0.92 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL5743785 0.92 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4942975 0.92 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4936174 0.92 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4940385 0.92 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4936543 0.92 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268419-A1 PYRROLIDINE DERIVATIVES USEFUL AS BAX INHIBITORS Applied Research Systems ARS Holding N.V. (AN) 2003-01-02 EP disclosed
WO-2001072705-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-04 WO disclosed