SCHEMBL7088046

SCHEMBL7088046

CO/N=C1\C[C@@H](C(=O)NC[C@@H](O)c2ccc(O)cc2)N(C(=O)c2ccc(-c3ccccc3OC)cc2)C1

nearest known ligand 0.76

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
OXTR P30559 5/20 0.76
AVPR1A P37288 3/20 0.76
FFAR2 O15552 14/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7089044 0.94 OXTR (0.85) OXTRAVPR1AFFAR2
SCHEMBL7081248 0.94 OXTR (0.85) OXTRAVPR1AFFAR2
SCHEMBL4939000 0.94 OXTR (0.85) OXTRAVPR1AFFAR2
SCHEMBL7083601 0.92 OXTR (0.70) OXTRAVPR1AFFAR2
SCHEMBL7083269 0.92 OXTR (0.70) OXTRAVPR1AFFAR2
SCHEMBL7090234 0.92 OXTR (0.70) OXTRAVPR1AFFAR2
SCHEMBL7087086 0.91 OXTR (0.90) OXTRAVPR1A
SCHEMBL7085545 0.86 OXTR (0.79) OXTRAVPR1AFFAR2
SCHEMBL7086784 0.86 OXTR (0.74) OXTRAVPR1A
SCHEMBL4943198 0.86 OXTR (1.00) OXTRAVPR1AFFAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268419-A1 PYRROLIDINE DERIVATIVES USEFUL AS BAX INHIBITORS Applied Research Systems ARS Holding N.V. (AN) 2003-01-02 EP disclosed
WO-2001072705-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-04 WO disclosed