SCHEMBL7081802

SCHEMBL7081802

CCC(O)c1nc(C(C)C)c(Sc2ccccc2)[nH]1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.39
LMNA P02545 1/20 0.37
GCGR P47871 3/20 0.35
RECQL P46063 1/20 0.32
SLC6A4 P31645 1/20 0.31
KDM4E B2RXH2 1/20 0.31
KMT2A Q03164 2/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30
MLKL Q8NB16 1/20 0.30
CXCL12 P48061 1/20 0.30
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7086217 0.86 DHFR (0.42) DHFRLMNASLC6A4KDM4EKMT2A
SCHEMBL7085415 0.85 TP53 (0.39) DHFRLMNASLC6A4KDM4EKMT2A
SCHEMBL7079967 0.85 GCGR (0.36) GCGR
SCHEMBL7078351 0.84 SLC6A4 (0.36) DHFRSLC6A4GAA
SCHEMBL7078733 0.83 HSP90B1 (0.32) DHFR
SCHEMBL6976919 0.83
SCHEMBL6963979 0.82 PTPRA (0.39) DHFRSLC6A4KDM4EKMT2A
SCHEMBL6961575 0.82 GCGR (0.32) GCGR
SCHEMBL7081085 0.81 RECQL (0.37) DHFRLMNARECQLSLC6A4KDM4E
SCHEMBL6974480 0.79 DHFR (0.34) DHFRKMT2AADORA2AADORA1CXCL12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed