SCHEMBL7083074

SCHEMBL7083074

Cc1ccc(N(CCc2cncn2Cc2ccc(C#N)cc2)C(C(N)=S)c2cccc(Cl)c2)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.44
CYP11B2 P19099 3/20 0.44
KCNH2 Q12809 3/20 0.44
FNTA P49354 12/20 0.43
FNTB P49356 12/20 0.43
PGGT1B P53609 6/20 0.42
NRAS P01111 1/20 0.42
HRAS P01112 1/20 0.42
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083071 0.79 KCNH2 (0.47) CYP11B1CYP11B2KCNH2FNTAFNTB
SCHEMBL7077067 0.77 CYP11B1 (0.45) CYP11B1CYP11B2KCNH2FNTAFNTB
SCHEMBL7083066 0.76 KCNH2 (0.47) CYP11B1CYP11B2KCNH2FNTAFNTB
SCHEMBL7083324 0.75 FNTA (0.49) CYP11B1CYP11B2KCNH2FNTAFNTB
SCHEMBL7085597 0.74 CYP11B1 (0.45) CYP11B1CYP11B2KCNH2FNTAFNTB
SCHEMBL7174102 0.73 CYP11B1 (0.47) CYP11B1CYP11B2KCNH2FNTAFNTB
SCHEMBL7083380 0.72 CYP11B1 (0.43) CYP11B1CYP11B2FNTAFNTB
SCHEMBL7078782 0.71 ALDH1A1 (0.45) CYP11B1CYP11B2FNTAFNTBPGGT1B
SCHEMBL7178460 0.71 FNTA (0.46) CYP11B1CYP11B2KCNH2FNTAFNTB
SCHEMBL7163852 0.71 FNTA (0.44) CYP11B1CYP11B2FNTAFNTBPGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1200430-A4 THIOUREA AND ISOTHIOUREA DERIVATIVES FOR INHIBITING RAS-TRANSFORMED CELL GROWTH YUHAN CORP LTD (KR) 2003-01-22 EP disclosed
EP-1200430-A1 THIOUREA AND ISOTHIOUREA DERIVATIVES FOR INHIBITING RAS-TRANSFORMED CELL GROWTH YUHAN CORPORATION, LTD. (KR) 2002-05-02 EP disclosed
WO-2001009128-A1 THIOUREA AND ISOTHIOUREA DERIVATIVES FOR INHIBITING RAS-TRANSFORMED CELL GROWTH YUHAN CORPORATION (KR) 2001-02-08 WO disclosed