SCHEMBL7085545

SCHEMBL7085545

CO/N=C1\C[C@@H](C(=O)NC[C@@H](O)c2ccc(O)c(OC)c2)N(C(=O)c2ccc(-c3ccccc3C)cc2)C1

nearest known ligand 0.79

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OXTR P30559 5/20 0.79
AVPR1A P37288 3/20 0.79
FFAR2 O15552 3/20 0.36
SLC22A3 O75751 1/20 0.36
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35
F2 P00734 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
ROCK2 O75116 3/20 0.34
ROCK1 Q13464 3/20 0.34
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7090234 0.95 OXTR (0.70) OXTRAVPR1AFFAR2SLC22A3F2
SCHEMBL7083601 0.95 OXTR (0.70) OXTRAVPR1AFFAR2SLC22A3F2
SCHEMBL7083269 0.90 OXTR (0.70) OXTRAVPR1AFFAR2
SCHEMBL7092416 0.89 OXTR (0.85) OXTRAVPR1AFFAR2TSHRROCK2
SCHEMBL4936354 0.89 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4940385 0.89 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4936174 0.89 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4942975 0.89 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4943198 0.89 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL5743785 0.89 OXTR (1.00) OXTRAVPR1AFFAR2ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268418-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS Applied Research Systems ARS Holding N.V. (AN) 2003-01-02 EP disclosed
WO-2001074769-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-11 WO disclosed