SCHEMBL7086519

SCHEMBL7086519

CCOC(=O)c1cc2cccc(OCCN3CCOCC3)c2o1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.56
CYP1A2 P05177 1/20 0.51
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
POLB P06746 1/20 0.47
CASP7 P55210 1/20 0.47
CASP6 P55212 1/20 0.47
CNR1 P21554 1/20 0.47
CNR2 P34972 1/20 0.47
KDM4E B2RXH2 4/20 0.47
HRH3 Q9Y5N1 1/20 0.46
ALDH1A1 P00352 2/20 0.46
PRKDC P78527 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MAPT P10636 1/20 0.46
PPARG P37231 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NCOR2 Q9Y618 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984399 0.91 KDM4E (0.56) RXFP1MEN1KMT2AKDM4EHRH3
SCHEMBL5564284 0.86 RXFP1 (0.59) RXFP1MEN1KMT2AL3MBTL1POLB
SCHEMBL3061600 0.79 LMNA (0.49) MEN1KMT2ACNR2ALDH1A1MAPT
SCHEMBL6982551 0.78 MAPK1 (0.49) CYP1A2MEN1KMT2ACNR2KDM4E
SCHEMBL4766909 0.78 CYP1A2 (0.62) CYP1A2CASP7CASP6KDM4EALDH1A1
SCHEMBL5559235 0.77 HRH3 (0.52) RXFP1MEN1KMT2APOLBKDM4E
SCHEMBL5558555 0.76 KDM4E (0.51) RXFP1MEN1KMT2APOLBKDM4E
SCHEMBL73410 0.76 LMNA (0.68) RXFP1MEN1KMT2AL3MBTL1POLB
SCHEMBL27297400 0.76 KMT2A (0.53) CYP1A2MEN1KMT2AL3MBTL1POLB
SCHEMBL5559654 0.76 RXFP1 (0.54) RXFP1MEN1KMT2APOLBCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1093367-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-03-05 EP claimed
EP-1093367-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-25 EP claimed
WO-1999066925-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-29 WO claimed
EP-1093367-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-03-05 EP disclosed
EP-1093367-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-25 EP disclosed
WO-1999066925-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-29 WO disclosed