SCHEMBL7086654

SCHEMBL7086654

CN1C(=O)C[C@H](c2ccccc2F)[C@@H]1C(=O)C(c1ccccc1)[C@H]1COC(=O)N1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 19/20 0.46
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6768415 0.70 HSD17B2 (0.39) HSD17B2ALDH1A1GAATSHR
SCHEMBL6768409 0.67 HSD17B2 (0.42) HSD17B2ALDH1A1GAATSHR
SCHEMBL6772387 0.67 HSD17B2 (0.42) HSD17B2ALDH1A1GAATSHR
SCHEMBL8882439 0.63 EPHX1 (0.39) HSD17B2
SCHEMBL11549245 0.63 EPHX1 (0.39) HSD17B2
SCHEMBL8882442 0.63 EPHX1 (0.39) HSD17B2
SCHEMBL12733121 0.63 ALDH1A1 (0.35) ALDH1A1GAA
SCHEMBL6768102 0.63 HSD17B2 (0.53) HSD17B2ALDH1A1GAATSHR
SCHEMBL6777855 0.63 HSD17B2 (0.53) HSD17B2ALDH1A1GAATSHR
SCHEMBL5182311 0.62 DAO (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1326829-A2 17-BETA-HYDROXYSTEROID DEHYDROGENASE-II INHIBITORS Bayer Pharmaceuticals Corporation (US) 2003-07-16 EP disclosed
WO-2002026706-A2 17-BETA-HYDROXYSTEROID DEHYDROGENASE-II INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2002-04-04 WO disclosed