SCHEMBL7088057

SCHEMBL7088057

COc1ccccc1Nc1n[nH]c(Sc2ccsc2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.44
MAPT P10636 7/20 0.44
ALDH1A1 P00352 6/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
KDM4E B2RXH2 2/20 0.44
KMT2A Q03164 2/20 0.44
GAA P10253 4/20 0.43
POLB P06746 3/20 0.43
PKM P14618 1/20 0.43
RECQL P46063 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HPGD P15428 2/20 0.41
IGF1R P08069 1/20 0.41
LRRK2 Q5S007 1/20 0.40
RAB9A P51151 5/20 0.40
ALOX15 P16050 2/20 0.40
HSD17B10 Q99714 2/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084013 0.82 ALDH1A1 (0.48) EGFRMAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL5371868 0.82 EGFR (0.41) EGFRMAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL7083252 0.81 EGFR (0.46) EGFRMAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL7084060 0.81 ALDH1A1 (0.44) EGFRMAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL6976057 0.80 MAPT (0.45) EGFRMAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL6980038 0.79 ALDH1A1 (0.45) EGFRMAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL7088181 0.79 GAA (0.48) MAPTALDH1A1SMN1; SMN2KDM4EKMT2A
SCHEMBL7090424 0.78 ALDH1A1 (0.49) EGFRMAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL7087949 0.78 EGFR (0.48) EGFRMAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL7083578 0.74 NPC1 (0.38) MAPTSMN1; SMN2KMT2ARAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1223932-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2003-01-15 EP disclosed
EP-1223932-A1 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2002-07-24 EP disclosed
WO-2001024796-A1 1,2,4-TRIAZOLE DERIVATIVES, COMPOSITION, PROCESS OF MAKING AND METHODS OF USE SMITHKLINE BEECHAM CORPORATION (US) 2001-04-12 WO disclosed