SCHEMBL7088461

SCHEMBL7088461

CC(C)c1nc2c([nH]1)c(=O)[nH]c(=O)n2Cc1cccc(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 3/20 0.50
PNP P00491 1/20 0.44
KDM4E B2RXH2 3/20 0.44
HPGD P15428 3/20 0.44
HTT P42858 3/20 0.44
LMNA P02545 1/20 0.44
GAA P10253 1/20 0.44
MEN1 O00255 1/20 0.44
PSMD14 O00487 1/20 0.44
TSHR P16473 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
POLB P06746 1/20 0.43
TRAP1 Q12931 2/20 0.43
HSP90B1 P14625 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
PDE9A O76083 2/20 0.42
PDE5A O76074 1/20 0.42
PDE1A P54750 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7090943 0.89 TLR7 (0.48) TLR7KDM4EHPGDHTTLMNA
SCHEMBL7676540 0.88 BRD4 (0.51) TLR7PNPHPGDGAAMEN1
SCHEMBL7090838 0.83 TLR7 (0.50) TLR7PNPKDM4EHPGDHTT
SCHEMBL6674800 0.78 PNP (0.54) PNPHTTMEN1KMT2ASMN1; SMN2
SCHEMBL7680197 0.77 TLR7 (0.48) TLR7HPGDHTTLMNAMEN1
SCHEMBL7426524 0.76 KMT2A (0.43) HPGDLMNAMEN1TSHRKMT2A
SCHEMBL11017605 0.75 ADORA2A (0.51) HPGDPOLBADORA2AADORA2BADORA1
SCHEMBL7092998 0.72 PDE4B (0.60)
SCHEMBL5226057 0.72 ADORA2A (0.56) HPGDADORA2AADORA2BADORA1
SCHEMBL7088426 0.72 TLR7 (0.48) TLR7TRAP1HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0814809-B1 ARYL THIOXANTHINES EURO CELTIQUE SA (LU) 2003-08-13 EP disclosed
US-6440979-B1 Aryl isoguanines EURO-CELTIQUE, S.A. (LU) 2002-08-27 US disclosed
US-6090816-A ANTIASTHMA AGENTS EURO-CELTIQUE S.A. (LU) 2000-07-18 US disclosed
US-6066641-A PHOSPHODIESTERASES AS MOLECULAR TARGETS FOR ANTI-ASTHMATIC AGENTS EURO-CELTIQUE S.A. (LU) 2000-05-23 US disclosed
WO-1996018399-A1 ARYL THIOXANTHINES EURO-CELTIQUE, S.A. (LU) 1996-06-20 WO disclosed