SCHEMBL7426524

SCHEMBL7426524

CC(C)c1nc2c([nH]1)c(=O)[nH]c(=O)n2CCCc1ccc(Cl)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.43
TSHR P16473 5/20 0.43
ALDH1A1 P00352 5/20 0.43
MEN1 O00255 4/20 0.43
HPGD P15428 4/20 0.43
MAPK1 P28482 2/20 0.43
RECQL P46063 1/20 0.43
MDM2 Q00987 1/20 0.43
XBP1 P17861 3/20 0.41
ATM Q13315 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TP53 P04637 2/20 0.41
USP2 O75604 2/20 0.41
HSD17B10 Q99714 2/20 0.41
DAO P14920 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
LMNA P02545 2/20 0.40
APOBEC3G Q9HC16 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7676540 0.87 BRD4 (0.51) KMT2ATSHRALDH1A1MEN1HPGD
SCHEMBL5226057 0.77 ADORA2A (0.56) HPGDHSD17B10ADORA2AADORA2B
SCHEMBL7088461 0.76 TLR7 (0.50) KMT2ATSHRALDH1A1MEN1HPGD
SCHEMBL7680197 0.76 TLR7 (0.48) KMT2ATSHRALDH1A1MEN1HPGD
SCHEMBL7090838 0.75 TLR7 (0.50) KMT2ATSHRMEN1HPGDADORA2A
SCHEMBL7416418 0.75 PDE4B (0.53) HSD17B10
SCHEMBL11017605 0.74 ADORA2A (0.51) HPGDHSD17B10ADORA2AADORA2BMAPT
SCHEMBL3229725 0.73 ADORA2A (0.47) ADORA2AADORA2B
SCHEMBL7091342 0.72 KDM4E (0.42) KMT2ATSHRALDH1A1MEN1HPGD
SCHEMBL7953405 0.71 ADORA2A (0.41) KMT2ATSHRALDH1A1MEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799040-A4 TRISUBSTITUTED THIOXANTHINES EURO CELTIQUE SA (LU) 1998-04-01 EP disclosed
EP-0799040-A1 TRISUBSTITUTED THIOXANTHINES Euroceltique S.A. (LU) 1997-10-08 EP disclosed
WO-1996018400-A1 TRISUBSTITUTED THIOXANTHINES EURO-CELTIQUE, S.A. (LU) 1996-06-20 WO disclosed