SCHEMBL7089030

SCHEMBL7089030

Fc1ccc(Nc2n[nH]c(Sc3ccco3)n2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 7/20 0.46
MAPT P10636 4/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
MAPK1 P28482 2/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
ALOX12 P18054 1/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
KDM4E B2RXH2 1/20 0.38
XBP1 P17861 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083129 0.88 GAA (0.49) KCNH3MAPTKMT2AMEN1MAPK1
SCHEMBL7084268 0.87 MAPT (0.46) MAPTKMT2AMEN1MAPK1NPC1
SCHEMBL5385724 0.80 KCNH3 (0.54) KCNH3MAPTKMT2AMEN1MAPK1
SCHEMBL7087516 0.79 NFKB1 (0.44) KCNH3MAPTKMT2AMEN1MAPK1
SCHEMBL7087949 0.75 EGFR (0.48) MAPTKMT2AMAPK1NPC1LMNA
SCHEMBL7083578 0.74 NPC1 (0.38) KCNH3MAPTKMT2AMEN1MAPK1
SCHEMBL7085921 0.73 CDC7 (0.38) KCNH3MAPTKMT2AMEN1MAPK1
SCHEMBL6985036 0.73 PDE4B (0.43) KCNH3MAPTKMT2AMEN1MAPK1
SCHEMBL7087741 0.73 CDK2 (0.43) KCNH3MAPTKMT2AMEN1MAPK1
SCHEMBL7090147 0.71 SYK (0.41) KCNH3MAPTKMT2AMEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1223932-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2003-01-15 EP disclosed
EP-1223932-A1 COMPOUNDS AND METHODS SmithKline Beecham Corporation (US) 2002-07-24 EP disclosed
WO-2001024796-A1 1,2,4-TRIAZOLE DERIVATIVES, COMPOSITION, PROCESS OF MAKING AND METHODS OF USE SMITHKLINE BEECHAM CORPORATION (US) 2001-04-12 WO disclosed