SCHEMBL7089158

SCHEMBL7089158

CNC(=O)C(C(C)c1ccc(Cl)cc1)C(C)c1ccc(Cl)cc1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FFAR2 O15552 5/20 0.64
ALDH1A1 P00352 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
PRCP P42785 3/20 0.44
BRD4 O60885 1/20 0.43
CNR1 P21554 1/20 0.42
ADRB2 P07550 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
MEN1 O00255 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7091260 0.81 HDAC3 (0.47) FFAR2ALDH1A1HDAC4HDAC7HDAC5
SCHEMBL26955949 0.81 FFAR2 (0.68) FFAR2ALDH1A1HDAC4HDAC7HDAC5
SCHEMBL1978851 0.79 HDAC4 (0.68) FFAR2ALDH1A1HDAC4HDAC7HDAC5
SCHEMBL25460815 0.78 FFAR2 (1.00) FFAR2MEN1KMT2A
SCHEMBL10949851 0.78 FFAR2 (1.00) FFAR2MEN1KMT2A
SCHEMBL13789274 0.77 FFAR2 (0.62) FFAR2ALDH1A1HDAC4HDAC7HDAC5
SCHEMBL3736159 0.76 FFAR2 (0.61) FFAR2ALDH1A1HDAC4HDAC7HDAC5
SCHEMBL20290805 0.76 FFAR2 (0.61) FFAR2ALDH1A1HDAC4HDAC7HDAC5
SCHEMBL11949354 0.72 ADRB2 (0.62) FFAR2HDAC4HDAC7HDAC5SLC6A4
SCHEMBL21430159 0.71 FFAR2 (0.56) FFAR2ALDH1A1HDAC4HDAC7HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322599-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-07-02 EP disclosed
WO-2001096283-A9 HIV INTEGRASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2002-10-17 WO disclosed
WO-2001096283-A2 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-12-20 WO disclosed