SCHEMBL7089530

SCHEMBL7089530

CS(=O)(=O)c1ccccc1-c1ccc(CNC(=O)CCc2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
L3MBTL1 Q9Y468 1/20 0.56
TRPV1 Q8NER1 2/20 0.54
ERCC1 P07992 1/20 0.51
ERCC4 Q92889 1/20 0.51
LTB4R2 Q9NPC1 1/20 0.51
SCN9A Q15858 3/20 0.49
PAX8 Q06710 1/20 0.48
LMNA P02545 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
GAA P10253 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
HDAC1 Q13547 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7091162 0.84 MAPT (0.58) ALDH1A1L3MBTL1LMNAGAAMEN1
SCHEMBL8792470 0.80 ALDH1A1 (0.71) ALDH1A1L3MBTL1TRPV1ERCC1ERCC4
SCHEMBL1661081 0.78 TRPV1 (0.76) ALDH1A1L3MBTL1TRPV1ERCC1ERCC4
SCHEMBL5299504 0.76 HCAR2 (0.53) ALDH1A1CYP2C9
SCHEMBL25046063 0.76 ALDH1A1 (0.71) ALDH1A1L3MBTL1TRPV1ERCC1ERCC4
SCHEMBL29171580 0.76 ALDH1A1 (0.71) ALDH1A1L3MBTL1TRPV1ERCC1ERCC4
SCHEMBL7030338 0.75 CA12 (0.67) ALDH1A1L3MBTL1TRPV1ERCC1ERCC4
SCHEMBL5177117 0.75 ALDH1A1 (0.66) ALDH1A1L3MBTL1TRPV1ERCC1ERCC4
SCHEMBL7600977 0.74 F10 (0.58) SCN9A
SCHEMBL1894742 0.74 TRPV1 (0.82) ALDH1A1L3MBTL1TRPV1ERCC1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1341755-A1 CARBOXYLIC ACID AMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF THROMBOEMBOLIC DISEASES AND TUMOURS MERCK PATENT GmbH (DE) 2003-09-10 EP disclosed
WO-2002048099-A1 CARBOXYLIC ACID AMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF THROMBOEMBOLIC DISEASES AND TUMOURS MERCK PATENT GMBH (DE) 2002-06-20 WO disclosed