SCHEMBL7089781

SCHEMBL7089781

CON=C1C[C@@H](C(=O)NC[C@@H](O)c2ccccc2)N(C(=O)c2ccc(-c3ccccc3)c(C(F)(F)F)c2)C1

nearest known ligand 0.75

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OXTR P30559 5/20 0.75
AVPR1A P37288 3/20 0.71
FFAR2 O15552 1/20 0.40
ROCK2 O75116 2/20 0.37
ROCK1 Q13464 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
S1PR1 P21453 1/20 0.35
PDK2 Q15119 3/20 0.34
SRD5A2 P31213 1/20 0.34
SCD O00767 3/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
MMP1 P03956 1/20 0.33
MMP3 P08254 1/20 0.33
MMP7 P09237 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4943344 0.92 OXTR (0.80) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL7078906 0.92 OXTR (0.80) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL7083271 0.89 OXTR (0.83) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL4945458 0.89 OXTR (0.83) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL7219611 0.88 OXTR (0.79) OXTRAVPR1AFFAR2ROCK2ROCK1
SCHEMBL4945256 0.86 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL4945247 0.86 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL4936262 0.86 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL4936835 0.86 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1
SCHEMBL4944776 0.86 OXTR (1.00) OXTRAVPR1AROCK2ROCK1MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268419-A1 PYRROLIDINE DERIVATIVES USEFUL AS BAX INHIBITORS Applied Research Systems ARS Holding N.V. (AN) 2003-01-02 EP disclosed
WO-2001072705-A1 PHARMACEUTICALLY ACTIVE PYRROLIDINE DERIVATIVES AS BAX INHIBITORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-10-04 WO disclosed