SCHEMBL7090429

SCHEMBL7090429

CC(C)(C)[C@@]1(OC(N)=O)CCCCN(Cc2ccccc2)C1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.49
MEN1 O00255 2/20 0.49
RIPK1 Q13546 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.41
TSHR P16473 2/20 0.40
CYP2D6 P10635 4/20 0.39
ALDH1A1 P00352 1/20 0.39
HCRTR1 O43613 2/20 0.39
HCRTR2 O43614 2/20 0.39
POLB P06746 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PREP P48147 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM3 P20309 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
OPRL1 P41146 1/20 0.37
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29048162 0.75 PTGDR2 (0.43) KMT2AL3MBTL1ALDH1A1CYP2C9CYP2C19
SCHEMBL29048193 0.69 PTGDR2 (0.42) KMT2AMEN1L3MBTL1ALDH1A1
SCHEMBL3188853 0.69 KMT2A (0.64) KMT2AMEN1RIPK1L3MBTL1TSHR
SCHEMBL1948718 0.68 KMT2A (0.52) KMT2AMEN1RIPK1L3MBTL1CYP2D6
SCHEMBL27699066 0.68 KMT2A (0.62) KMT2AMEN1RIPK1L3MBTL1TSHR
SCHEMBL28702537 0.68 RXFP1 (0.34) KMT2AALDH1A1HRH3
SCHEMBL9726979 0.67 KMT2A (1.00) KMT2AMEN1RIPK1L3MBTL1TSHR
SCHEMBL29048188 0.67 MT-CO2 (0.39) KMT2AMEN1ALDH1A1CYP2C9CYP2C19
SCHEMBL19641147 0.66 CYP2D6 (0.55) TSHRCYP2D6ALDH1A1POLBCYP2C9
SCHEMBL835093 0.66 KMT2A (0.64) KMT2AMEN1RIPK1L3MBTL1HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294716-A1 LACTAM INHIBITORS OF FACTOR XA AND METHOD Bristol-Myers Squibb Company (US) 2003-03-26 EP disclosed
WO-2001096331-A1 LACTAM INHIBITORS OF FACTOR XA AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 2001-12-20 WO disclosed